SCHEMBL4178461

SCHEMBL4178461

Nc1ccc(N2CCN(C(=O)CO)CC2)cc1OC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.46
ALK Q9UM73 5/20 0.46
EGFR P00533 1/20 0.44
POLB P06746 2/20 0.44
ENPP2 Q13822 3/20 0.41
ME2 P23368 1/20 0.41
ME1 P48163 1/20 0.41
ME3 Q16798 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
CCR1 P32246 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11344943 0.86 IP6K1 (0.43) LMNAHTT
SCHEMBL4181229 0.85 CASP6 (0.54) ALKEGFRENPP2MAPT
SCHEMBL2723108 0.84 ALK (0.53) AKR1C3ALKALDH1A1LMNAMAPT
SCHEMBL2724815 0.81 MAPT (0.54) ALKEGFRALDH1A1LMNAMAPT
SCHEMBL29673386 0.79 MAPT (0.46) POLBALDH1A1KDM4ELMNAGAA
SCHEMBL29771877 0.78 GAA (0.56) ALDH1A1KDM4EGAAMAPTHTT
SCHEMBL409735 0.78 GAA (0.56) ALDH1A1KDM4EGAAMAPTHTT
Hydrochloric Acid SCHEMBL3502999 0.77 MAPT (0.55) ALDH1A1KDM4EGAAMAPTHTT
SCHEMBL27925817 0.76 CREBBP (0.36) ALDH1A1KDM4ELMNAGAAMAPT
SCHEMBL13362063 0.75 MAPT (0.58) POLBALDH1A1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061299-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2012-05-10 WO disclosed