SCHEMBL41795

SCHEMBL41795

CC1(C)CC(c2cccc(N3CCOCC3)c2)Nc2ccc(C(=O)NCCN3CCSCC3(O)O)cc21

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NTRK1 P04629 2/20 0.35
NTRK3 Q16288 1/20 0.35
NTRK2 Q16620 1/20 0.35
DRD4 P21917 2/20 0.34
HTR1A P08908 1/20 0.34
CYP2C19 P33261 3/20 0.34
POLB P06746 2/20 0.34
CYP2C9 P11712 1/20 0.34
MAPT P10636 1/20 0.34
DRD3 P35462 2/20 0.34
HDAC3 O15379 1/20 0.34
PARP1 P09874 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL42389 0.90 HDAC4 (0.36) HSD17B10DRD4HTR1APOLBMAPT
SCHEMBL45313 0.85 PRKD1 (0.40) MEN1RAB9AKMT2AHSD17B10NTRK1
SCHEMBL45394 0.85 PRKD1 (0.40) MEN1RAB9AKMT2AHSD17B10NTRK1
SCHEMBL45444 0.83 HSD17B10 (0.42) MEN1RAB9AKMT2AHSD17B10DRD4
SCHEMBL45445 0.83 HSD17B10 (0.42) MEN1RAB9AKMT2AHSD17B10DRD4
SCHEMBL11026483 0.81 F10 (0.45) MEN1KMT2ANTRK1NTRK3NTRK2
SCHEMBL45257 0.80 PRMT5 (0.44) MEN1RAB9AKMT2ANTRK1NTRK3
SCHEMBL45312 0.79 F10 (0.47) CYP2C19CYP2C9MAPTHDAC3CYP1A2
SCHEMBL45003 0.79 F10 (0.39) NTRK1NTRK3NTRK2CYP2C19MAPT
SCHEMBL41549 0.78 KMO (0.52) MEN1KMT2AHSD17B10CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588458-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-08 EP claimed
WO-2012001020-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-05 WO claimed