Danofloxacin

Danofloxacin

SCHEMBL418388

CN1C[C@@H]2C[C@H]1CN2c1cc2c(cc1F)c(=O)c(C(=O)O)cn2C1CC1.CS(=O)(=O)O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Danofloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG known ✓ P48736 5/20 0.47
PIK3CD known ✓ O00329 3/20 0.47
PIK3R1 known ✓ P27986 3/20 0.47
PIK3CA known ✓ P42336 3/20 0.47
KDM4E B2RXH2 5/20 0.57
ALDH1A1 P00352 5/20 0.57
LMNA P02545 3/20 0.56
HPGD P15428 3/20 0.56
HSD17B10 Q99714 2/20 0.56
CYP1A2 P05177 1/20 0.56
TOP2A P11388 1/20 0.56
CYP2C9 P11712 1/20 0.56
TOP2B Q02880 1/20 0.56
MAPT P10636 1/20 0.56
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Danofloxacin SCHEMBL30014294 1.00 KDM4E (0.57) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL149627 0.95 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL9669908 0.95 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL10073753 0.95 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL29658817 0.95 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL16518619 0.95 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL28372629 0.94 KDM4E (0.61) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL31592056 0.94 KDM4E (0.54) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9670553 0.90 KDM4E (0.63) KDM4EALDH1A1LMNAHPGDHSD17B10
Danofloxacin SCHEMBL31592064 0.89 KDM4E (0.59) KDM4EALDH1A1LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 346 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118191116-A Method for detecting illegally added medicines in eucommia ulmoides leaf extract 山东省饲料兽药质量检验中心 2024-06-14 CN claimed
CN-114191566-B Method for preparing ZIF-8 composite nano material with magnetic targeting, antibacterial and developing functions 上海交通大学 2023-09-29 CN claimed
CN-115368369-A Synthesis method of demethylation impurity of danofloxacin mesylate 浙江国邦药业有限公司 2022-11-22 CN claimed
CN-110060784-B Drug resistance judgment standard test method for mycoplasma gallisepticum to danofloxacin 华中农业大学 2022-11-08 CN claimed
US-20220249473-A1 A NOVEL THERAPY FOR ERYTHROPOIETIC PROTOPORPHYRIA (EPP) AND X-LINKED PROTOPORPHYRIA (XLP) UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2022-08-11 US claimed
EP-3972605-A1 A NOVEL THERAPY FOR ERYTHROPOIETIC PROTOPORPHYRIA (EPP) AND X-LINKED PROTOPORPHYRIA (XLP) University of Pittsburgh - of the Commonwealth System of Higher Education (US) 2022-03-30 EP claimed
CN-114191566-A Method for preparing ZIF-8 composite nano material with magnetic targeting, antibacterial and developing functions 上海交通大学 2022-03-18 CN claimed
CN-114105999-A Synthesis method of danofloxacin mesylate 浙江国邦药业有限公司 2022-03-01 CN claimed
CN-114096250-A Novel therapy for erythropoietic protoporphyrinopathy (EPP) and X-linked protoporphyrinopathy (XLP) 匹兹堡大学联邦高等教育系统 2022-02-25 CN claimed
CN-114010797-A Bacteria-targeted nano antibacterial agent and preparation method thereof 上海交通大学 2022-02-08 CN claimed
CN-101703469-A Preparation method and products of danofloxacin mesylate liposome UNIV NORTHEAST AGRICULTURAL 2010-05-12 CN claimed
WO-2009088831-A2 METHOD OF INHIBITING ABCG2 AND OTHER TREATMENT METHODS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2009-07-16 WO claimed
WO-2009061770-A2 METHOD OF INHIBITING ABCG2 AND RELATED TREATMENTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2009-05-14 WO claimed
CN-101411689-A Danofloxacin mesylate microsphere formulation for livestock and poultry and preparation method thereof HUBEI PIG VETERINARY MEDICINE (CN) 2009-04-22 CN claimed
EP-1656018-A4 EDIBLE FILMS FOR ADMINISTRATION OF MEDICAMENTS TO ANIMALS INNOZEN INC (US) 2008-07-23 EP claimed
CN-1965828-A Dafloxacin mesylate solution containing hexacyclic ring water for animals TIANJIN RINGTOP BIOTECHNOLOGY (CN) 2007-05-23 CN claimed
EP-1656018-A1 EDIBLE FILMS FOR ADMINISTRATION OF MEDICAMENTS TO ANIMALS Innozen, Inc. (US) 2006-05-17 EP claimed
US-20050136096-A1 Edible films for administration of medicaments to animals, methods for their manufacture and methods for their use for the treatment of animals CUREX PHARMACEUTICAL MEXICO S.A.P.I. DE C.V. (MX) 2005-06-23 US claimed
WO-2005018323-A1 EDIBLE FILMS FOR ADMINISTRATION OF MEDICAMENTS TO ANIMALS INNOZEN, INC. (US) 2005-03-03 WO claimed
US-4861779-A Anti-bacterial substituted bridged-diazabicycloalkyl quinolone carboxylic acids PFIZER INC. (US) 1989-08-29 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220249473-A1 A NOVEL THERAPY FOR ERYTHROPOIETIC PROTOPORPHYRIA (EPP) AND X-LINKED PROTOPORPHYRIA (XLP) XPA, TPX2, XPOT PIK3CG 3451/4885PIK3CD 3690/4885PIK3R1 4008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.