SCHEMBL4184437

SCHEMBL4184437

COc1ccc(-c2cncc(NCc3ccc(Cl)cc3)c2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 5/20 0.51
KCNH2 Q12809 1/20 0.50
PDE4B Q07343 1/20 0.47
KIT P10721 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
PRKCQ Q04759 1/20 0.46
MAPK1 P28482 2/20 0.46
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PLK1 P53350 1/20 0.45
HPGD P15428 1/20 0.45
DYRK1A Q13627 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4189065 0.90 ALDH1A1 (0.56) KCNH2PDE4BMEN1KMT2ALMNA
SCHEMBL4180512 0.86 KCNH2 (0.51) KCNH2PDE4BMEN1KMT2ALMNA
SCHEMBL4196517 0.84 DYRK1A (0.54) KCNH2PDE4BMAPTDYRK1ACLK4
SCHEMBL4930981 0.81 CNR1 (0.49) ALPLKCNH2PDE4BMEN1KMT2A
SCHEMBL4187573 0.81 FYN (0.61) ALPLKCNH2KITKMT2ALMNA
SCHEMBL4155473 0.81 ALDH1A1 (0.51) KCNH2MEN1KMT2ALMNAL3MBTL1
SCHEMBL4189975 0.80 FYN (0.55) KCNH2PDE4BKMT2ALMNAL3MBTL1
SCHEMBL4191630 0.80 ALDH1A1 (0.53) ALPLKCNH2PDE4BKITKMT2A
SCHEMBL4189206 0.80 MAPT (0.58) KITMEN1KMT2AMAPK1LMNA
SCHEMBL4187548 0.78 SCN10A (0.47) ALPLMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090196912-A1 Pyridinylamines GPC BOTECH AG (DE) 2009-08-06 US claimed
EP-1789393-A2 PYRIDINYLAMINES GPC Biotech AG (DE) 2007-05-30 EP claimed
WO-2006010637-A2 PYRIDINYLAMINES GPC BIOTECH AG (DE) 2006-02-02 WO claimed
US-20200206188-A1 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF INDIRUBIN AND ANALOGS THEREOF, INCLUDING MEISOINDIGO BROWN DENNIS M (US) 2020-07-02 US disclosed
US-10383847-B2 Compositions and methods to improve the therapeutic benefit of indirubin and analogs thereof, including meisoindigo BROWN DENNIS M (US) 2019-08-20 US disclosed
US-20160243077-A1 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF INDIRUBIN AND ANALOGS THEREOF, INCLUDING MEISOINDIGO BROWN DENNIS M (US) 2016-08-25 US disclosed
US-20090196912-A1 Pyridinylamines GPC BOTECH AG (DE) 2009-08-06 US disclosed
EP-1789393-A2 PYRIDINYLAMINES GPC Biotech AG (DE) 2007-05-30 EP disclosed
WO-2006010637-A2 PYRIDINYLAMINES GPC BIOTECH AG (DE) 2006-02-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10383847-B2 Compositions and methods to improve the therapeutic benefit of indirubin and analogs thereof, including meisoindigo NEK9, NEK7, NEK3 ALPL 1226/4885KCNH2 3526/4885PDE4B 2776/4885
US-20200206188-A1 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF INDIRUBIN AND ANALOGS THEREOF, INCLUDING MEISOINDIGO NEK9, NEK7, NEK3 ALPL 1226/4885KCNH2 3526/4885PDE4B 2776/4885
US-20160243077-A1 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF INDIRUBIN AND ANALOGS THEREOF, INCLUDING MEISOINDIGO NEK9, NEK7, NEK3 ALPL 1226/4885KCNH2 3526/4885PDE4B 2776/4885
US-20090196912-A1 Pyridinylamines PRNP, PLPBP, SNCA ALPL 2140/4885KCNH2 763/4885PDE4B 709/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.