SCHEMBL4186249

SCHEMBL4186249

Fc1ccc(-c2nc(=S)[nH][nH]2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.66
GAA P10253 7/20 0.66
KDM4E B2RXH2 7/20 0.66
HPGD P15428 6/20 0.66
APOBEC3G Q9HC16 5/20 0.66
ALOX12 P18054 3/20 0.66
PKM P14618 1/20 0.66
GFER P55789 5/20 0.65
DCUN1D1 Q96GG9 7/20 0.64
MPI P34949 6/20 0.59
TDP1 Q9NUW8 4/20 0.59
RAB9A P51151 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
ALOX15 P16050 2/20 0.54
HSD17B10 Q99714 2/20 0.54
NPSR1 Q6W5P4 1/20 0.54
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
RXFP1 Q9HBX9 1/20 0.50
QPCT Q16769 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17541734 0.79 GFER (1.00) ALDH1A1GAAKDM4EHPGDAPOBEC3G
SCHEMBL7996480 0.67 ALDH1A1 (0.44) ALDH1A1GAAKDM4EHPGDAPOBEC3G
SCHEMBL7622866 0.64 MAPK1 (0.47) ALDH1A1KDM4EHPGDGFERRAB9A
SCHEMBL24317550 0.64 NPC1 (0.47) ALDH1A1GAAKDM4EHPGDPKM
SCHEMBL15029205 0.62 MAPK1 (0.42) ALDH1A1GAAKDM4EPKMRAB9A
SCHEMBL15007066 0.62 NR1H2 (0.64) ALDH1A1HPGDRAB9ASMN1; SMN2LMNA
SCHEMBL11838228 0.62 KDM4E (0.50) ALDH1A1GAAKDM4EHPGDPKM
SCHEMBL12562793 0.61 BCL2L1 (0.55) RAB9ASMN1; SMN2POLB
SCHEMBL10337645 0.61 BCL2L1 (0.55) RAB9ASMN1; SMN2POLB
SCHEMBL197346 0.61 BCL2L1 (0.55) RAB9ASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009087218-A1 THIAZOLTRIAZOLES AND THIAZOLIMIDAZOLES AS ANTAGONISTS OF THE MGLUR5 RECEPTOR GLAXO GROUP LIMITED (GB) 2009-07-16 WO disclosed