SCHEMBL4188897

SCHEMBL4188897

Cc1ccc(C)c(-c2cnc(N)nc2N)c1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.54
FGFR1 P11362 1/20 0.49
ADORA1 P30542 1/20 0.44
LCK P06239 1/20 0.41
KDR P35968 1/20 0.41
JAK3 P52333 1/20 0.41
MAPK14 Q16539 1/20 0.41
RPS6KA3 P51812 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4357670 0.86 DHFR (0.50) DHFRFGFR1ADORA1LCKKDR
SCHEMBL1612609 0.83 DHFR (0.51) DHFRFGFR1LCKKDRJAK3
SCHEMBL27612441 0.80 DHFR (0.55) DHFRFGFR1ADORA1LCKKDR
SCHEMBL4464780 0.79 FGFR1 (0.55) DHFRFGFR1ADORA1LCKKDR
SCHEMBL736022 0.77 DHFR (0.58) DHFRFGFR1ADORA1RPS6KA3
SCHEMBL4486186 0.75 FGFR1 (0.55) DHFRFGFR1ADORA1LCKKDR
SCHEMBL1388276 0.75 ADORA1 (0.70) DHFRFGFR1ADORA1LCKKDR
SCHEMBL27631706 0.75 DHFR (0.68) DHFRFGFR1ADORA1LCKKDR
SCHEMBL30488016 0.75 ADORA1 (0.70) DHFRFGFR1ADORA1LCKKDR
SCHEMBL4200127 0.73 FGFR1 (0.71) DHFRFGFR1ADORA1LCKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032543-A1 2-ANILINO-4-AMINOALKYLENEAMINOPYRIMIDINES Boehringer Ingelheim International GmbH (DE) 2009-03-11 EP disclosed
WO-2007146977-A1 2-ANILINO-4-AMINOALKYLENEAMINOPYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-12-21 WO disclosed