SCHEMBL4189264

SCHEMBL4189264

Cc1nc(NC(=O)c2ccco2)sc1C(=O)O.NC(=O)c1ccc(Cl)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.76
TDP1 Q9NUW8 1/20 0.76
ALDH1A1 P00352 4/20 0.61
HPGD P15428 4/20 0.61
ADORA3 P0DMS8 3/20 0.61
LCK P06239 2/20 0.58
RAB9A P51151 8/20 0.58
KDM4E B2RXH2 4/20 0.58
NPC1 O15118 7/20 0.56
NPSR1 Q6W5P4 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
MAPT P10636 4/20 0.56
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
LMNA P02545 3/20 0.56
POLB P06746 1/20 0.56
TSHR P16473 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.53
ADORA2A P29274 2/20 0.53
ADORA1 P30542 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4189293 0.90 PKM (0.76) PKMTDP1ALDH1A1HPGDADORA3
SCHEMBL3587905 0.87 PKM (1.00) PKMTDP1ALDH1A1HPGDADORA3
SCHEMBL4197928 0.85 NPC1 (0.67) PKMTDP1ALDH1A1HPGDADORA3
SCHEMBL4195677 0.83 PKM (0.70) PKMTDP1ALDH1A1HPGDLCK
SCHEMBL4349298 0.81 NPC1 (0.65) PKMTDP1ALDH1A1ADORA3LCK
SCHEMBL4915021 0.80 NPC1 (0.63) PKMTDP1ALDH1A1LCKRAB9A
SCHEMBL4346190 0.80 NPC1 (0.80) PKMTDP1ALDH1A1ADORA3LCK
SCHEMBL4397896 0.79 PKM (0.83) PKMTDP1ALDH1A1HPGDADORA3
SCHEMBL3587473 0.76 KDM4E (0.81) PKMTDP1ALDH1A1HPGDADORA3
SCHEMBL4187284 0.76 NPC1 (0.52) ALDH1A1ADORA3LCKRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029138-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2009-03-04 EP claimed
WO-2007130075-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-11-15 WO claimed