Terephthalamide

Terephthalamide

SCHEMBL4193901

NC(=O)c1ccc(C(N)=O)cc1.NC(=O)c1cccc(C(N)=O)c1.NCCN

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Terephthalamide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.57
PARP10 Q53GL7 5/20 0.56
PARP15 Q460N3 3/20 0.56
PARP14 Q460N5 2/20 0.56
TNKS O95271 1/20 0.56
TNKS2 Q9H2K2 1/20 0.56
PARP2 Q9UGN5 1/20 0.56
TSHR P16473 2/20 0.56
POLB P06746 1/20 0.56
CYP3A4 P08684 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C19 P33261 1/20 0.56
RECQL P46063 1/20 0.56
BLM P54132 1/20 0.56
PMP22 Q01453 1/20 0.56
HSD17B10 Q99714 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
KIF11 P52732 2/20 0.49
PLA2G10 O15496 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethylenediamine SCHEMBL6068910 0.96 PARP1 (0.61) PARP1PARP10PARP15PARP14TNKS
Terephthalamide SCHEMBL5692322 0.91 PARP1 (0.67) PARP1PARP10PARP15PARP14TNKS
Terephthalamide SCHEMBL704245 0.90 PARP1 (0.52) PARP1PARP10PARP15PARP14TNKS
SCHEMBL10458793 0.89 PARP1 (0.64) PARP1PARP10PARP15PARP14TNKS
SCHEMBL31021028 0.86 PARP1 (0.73) PARP1PARP10PARP15PARP14TNKS
SCHEMBL36694 0.86 PARP1 (0.73) PARP1PARP10PARP15PARP14TNKS
SCHEMBL294705 0.85 PARP1 (0.55) PARP1PARP10PARP15PARP14TNKS
Terephthalamide SCHEMBL4985044 0.84 PARP1 (0.59) PARP1PARP10PARP15PARP14TNKS
Water SCHEMBL7768285 0.84 PARP1 (0.70) PARP1PARP10PARP15PARP14TNKS
Methane SCHEMBL688609 0.84 PARP1 (0.70) PARP1PARP10PARP15PARP14TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1769028-A4 GAS-BARRIER NANOCOMPOSITE COMPOSITION AND ARTICLE USING THE SAME LG CHEMICAL LTD (KR) 2009-03-11 EP disclosed
EP-1769028-A1 GAS-BARRIER NANOCOMPOSITE COMPOSITION AND ARTICLE USING THE SAME LG Chem. Ltd. (KR) 2007-04-04 EP disclosed
WO-2006009360-A1 GAS-BARRIER NANOCOMPOSITE COMPOSITION AND ARTICLE USING THE SAME LG CHEM. LTD. (KR) 2006-01-26 WO disclosed