SCHEMBL4196133

SCHEMBL4196133

COc1cc(NC(=O)c2cccc3ccccc23)c(C(=O)NCC2CCCCC2)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 9/20 0.69
CNR2 P34972 8/20 0.69
AURKA O14965 1/20 0.53
LCK P06239 1/20 0.53
MET P08581 1/20 0.53
KDR P35968 1/20 0.53
TEK Q02763 1/20 0.53
AURKB Q96GD4 1/20 0.53
NPC1 O15118 2/20 0.52
ALDH1A1 P00352 2/20 0.52
BCHE P06276 1/20 0.48
PDE10A Q9Y233 1/20 0.48
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GAA P10253 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224036 0.87 CNR1 (0.74) CNR1CNR2AURKALCKMET
SCHEMBL4199022 0.83 CNR1 (0.64) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL5224040 0.82 CNR1 (0.78) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL5314765 0.82 CNR1 (0.78) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4190780 0.82 CNR1 (1.00) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4190849 0.82 CNR1 (0.78) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL5220662 0.82 CNR1 (0.74) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4194677 0.81 CNR1 (0.73) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4191810 0.79 CNR1 (0.73) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4185327 0.79 CNR1 (0.73) CNR1CNR2NPC1ALDH1A1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP claimed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO claimed
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP disclosed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO disclosed