SCHEMBL4196376

SCHEMBL4196376

[CH2]C(OC)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.44
IDO1 P14902 2/20 0.43
TDO2 P48775 2/20 0.43
SLC6A3 Q01959 3/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
ACHE P22303 1/20 0.36
NFE2L2 Q16236 1/20 0.34
HTT P42858 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
CHRM1 P11229 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
HRH1 P35367 1/20 0.33
CYP17A1 P05093 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10813004 0.78 CHRNA7 (0.41) ACHENFE2L2ALDH1A1MAPT
SCHEMBL16798345 0.76 CA1 (0.52) AOC3ACHEHTTALDH1A1MAPT
SCHEMBL16798444 0.76 SLC6A4 (0.48) AOC3IDO1TDO2SLC6A3SLC6A2
SCHEMBL28835630 0.76 TDP1 (0.42) ACHEALDH1A1MAPTTSHRMAPK1
SCHEMBL16952921 0.76 CES2 (0.38) SLC6A4NFE2L2ALDH1A1MAPTCYP2C19
SCHEMBL7327576 0.75 KMT2A (0.41) CYP2D6TSHRHRH1LMNA
SCHEMBL6205426 0.75 AOC3 (0.47) AOC3IDO1TDO2SLC6A3SLC6A2
SCHEMBL792136 0.75 IDO1 (0.58) AOC3IDO1TDO2SLC6A3SLC6A2
SCHEMBL27238 0.75 KMT2A (0.41) CYP2D6TSHRHRH1LMNA
SCHEMBL16950984 0.74 AOC3 (0.50) AOC3IDO1TDO2ACHENFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1034501-C (Bemzhydryloxyethylpiperidyl) aliphatic acid derivatives and their use in the treatment of allergies and asthma SANKYO CO (JP) 1997-04-09 CN claimed
CN-1058773-A (diphenyl-methyl oxyethyl group piperidyl) aliphatic acid derivative and the purposes in treatment allergy and asthma thereof SANKYO CO (JP) 1992-02-19 CN claimed
EP-1796675-A4 COMPOSITIONS AND METHODS FOR TREATING OPHTHALMIC DISEASES MERCK & CO INC (US) 2009-03-04 EP disclosed
EP-1796675-A2 COMPOSITIONS AND METHODS FOR TREATING OPHTHALMIC DISEASES Merck & Co., Inc. (US) 2007-06-20 EP disclosed
WO-2006039252-A2 COMPOSITIONS AND METHODS FOR TREATING OPHTHALMIC DISEASES MERCK & CO., INC. (US) 2006-04-13 WO disclosed
EP-0906308-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES AS 5-HT1D RECEPTOR AGONISTS MERCK SHARP & DOHME LTD. (GB) 1999-04-07 EP disclosed
EP-0861244-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1998-09-02 EP disclosed
WO-1997045426-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES AS 5-HT1D RECEPTOR AGONISTS MERCK SHARP & DOHME LIMITED (GB) 1997-12-04 WO disclosed
EP-0804434-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1997-11-05 EP disclosed
WO-1997018201-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1997-05-22 WO disclosed
CN-1034501-C (Bemzhydryloxyethylpiperidyl) aliphatic acid derivatives and their use in the treatment of allergies and asthma SANKYO CO (JP) 1997-04-09 CN disclosed
WO-1996004274-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1996-02-15 WO disclosed
CN-1058773-A (diphenyl-methyl oxyethyl group piperidyl) aliphatic acid derivative and the purposes in treatment allergy and asthma thereof SANKYO CO (JP) 1992-02-19 CN disclosed