Ganetespib

Ganetespib

SCHEMBL419750

CC(C)c1cc(-c2n[nH]c(=O)n2-c2ccc3c(ccn3C)c2)c(O)cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HSP90AA1HSP90AB1

The experimentally established mechanism targets of Ganetespib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AB1 known ✓ P08238 20/20 1.00
HSP90AA1 known ✓ P07900 18/20 1.00
HSP90B1 P14625 1/20 1.00
TRAP1 Q12931 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ganetespib SCHEMBL29352120 1.00 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
Ganetespib SCHEMBL29376128 1.00 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL501479 0.91 HSP90AB1 (0.82) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL9924656 0.89 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL500866 0.89 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL4566976 0.89 HSP90AB1 (0.79) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL4566979 0.89 HSP90AB1 (0.79) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL25602985 0.88 HSP90AB1 (0.78) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL419168 0.88 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL421109 0.88 HSP90AB1 (0.78) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 251 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250160275-A1 COMPOUNDS FOR MODIFYING MEIOTIC RECOMBINATION AND METHODS RELATING THERETO THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2025-05-22 US claimed
WO-2023164606-A1 COMPOUNDS FOR MODIFYING MEIOTIC RECOMBINATION AND METHODS RELATING THERETO THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2023-08-31 WO claimed
WO-2016073669-A1 COMBINATION THERAPY OF HSP90 INHIBITORY COMPOUNDS WITH MTOR INHIBITORS VUKOVIC VOJO (US) 2016-05-12 WO claimed
WO-2014018862-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING A HEAT SHOCK PROTEIN INHIBITOR AND A|PURINE DE NOVO SYNTHESIS INHIBITOR FOR TREATING RHEUMATOID ARTHRITIS OR CANCER CORNING INCORPORATED (US) 2014-01-30 WO claimed
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms KARTOS THERAPEUTICS INC (US) 2026-04-09 US disclosed
US-20250387383-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS KARTOS THERAPEUTICS, INC. (US) 2025-12-25 US disclosed
US-20250340615-A1 NOVEL FUSION MOLECULES AND USES THEREOF FOUNDATION MEDICINE, INC. (US) 2025-11-06 US disclosed
US-20250333479-A1 NOVEL FUSION MOLECULES AND USES THEREOF FOUNDATION MEDICINE, INC. (US) 2025-10-30 US disclosed
US-20250333480-A1 FUSION MOLECULES AND USES THEREOF FOUNDATION MEDICINE, INC. (US) 2025-10-30 US disclosed
EP-4629993-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS Kartos Therapeutics (US) 2025-10-15 EP disclosed
US-12378302-B2 Fusion molecules and uses thereof FOUNDATION MEDICINE, INC. (US) 2025-08-05 US disclosed
CN-120136941-A Anti-aging composition and application thereof 鲁贝多生命科学公司 2025-06-13 CN disclosed
US-20080027047-A1 Compounds that modulate HSP90 activity and methods for identifying same SYNTA PHARMACEUTICALS CORP 2008-01-31 US disclosed
US-20080027047-A1 Compounds that modulate HSP90 activity and methods for identifying same SYNTA PHARMACEUTICALS CORP 2008-01-31 US disclosed
US-20080004276-A1 Method for treating non-hodgkin's lymphoma LSI FINANCING LLC, AS ADMINISTRATIVE AGENT 2008-01-03 US disclosed
US-20080004276-A1 Method for treating non-hodgkin's lymphoma LSI FINANCING LLC, AS ADMINISTRATIVE AGENT 2008-01-03 US disclosed
US-20080004266-A1 Method for treating proliferative disorders associated with protooncogene products LSI FINANCING LLC, AS ADMINISTRATIVE AGENT 2008-01-03 US disclosed
US-20080004266-A1 Method for treating proliferative disorders associated with protooncogene products LSI FINANCING LLC, AS ADMINISTRATIVE AGENT 2008-01-03 US disclosed
WO-2007139960-A2 COMPOUNDS THAT MODULATE HSP90 ACTIVITY AND METHODS FOR IDENTIFYING SAME SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO disclosed
WO-2007139952-A2 METHOD FOR THE PREPARATION OF TRIAZOLE COMPOUNDS WITH HSP90 MODULATING ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250387383-A1 METHODS OF TREATING MYELOPROLIFERATIVE NEOPLASMS JAK2, JAK1, MPL HSP90AB1 303/4885HSP90AA1 392/4885HSP90B1 637/4885
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms JAK2, TP53, CDKN1A HSP90AB1 233/4885HSP90AA1 291/4885HSP90B1 593/4885
US-20250340615-A1 NOVEL FUSION MOLECULES AND USES THEREOF RPS27A, CD2BP2, FGB HSP90AB1 1029/4885HSP90AA1 1729/4885HSP90B1 172/4885
US-20080004276-A1 Method for treating non-hodgkin's lymphoma HSP90AB1, HSP90AB2P, HSP90B1 HSP90AB1 1/4885HSP90AA1 4/4885HSP90B1 3/4885
US-12378302-B2 Fusion molecules and uses thereof RPS27A, CD2BP2, FGB HSP90AB1 1053/4885HSP90AA1 1857/4885HSP90B1 138/4885
US-20250333479-A1 NOVEL FUSION MOLECULES AND USES THEREOF RPS27A, CD2BP2, FGB HSP90AB1 1029/4885HSP90AA1 1729/4885HSP90B1 172/4885
US-20080027047-A1 Compounds that modulate HSP90 activity and methods for identifying same HSP90AB1, HSP90B1, CDC37 HSP90AB1 1/4885HSP90AA1 4/4885HSP90B1 2/4885
US-20080004266-A1 Method for treating proliferative disorders associated with protooncogene products HSP90AB1, HSP90AB2P, HSP90AA1 HSP90AB1 1/4885HSP90AA1 3/4885HSP90B1 7/4885
US-20250333480-A1 FUSION MOLECULES AND USES THEREOF RPS27A, CD2BP2, FGB HSP90AB1 1053/4885HSP90AA1 1857/4885HSP90B1 138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.