Ganetespib

Ganetespib

SCHEMBL29352120

CC(C)c1cc(-c2n[nH]c(=O)n2-c2ccc3c(ccn3C)c2)c(O)cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HSP90AA1HSP90AB1

The experimentally established mechanism targets of Ganetespib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AB1 known ✓ P08238 20/20 1.00
HSP90AA1 known ✓ P07900 18/20 1.00
HSP90B1 P14625 1/20 1.00
TRAP1 Q12931 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ganetespib SCHEMBL419750 1.00 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
Ganetespib SCHEMBL29376128 1.00 HSP90AB1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL501479 0.91 HSP90AB1 (0.82) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL9924656 0.89 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL500866 0.89 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL4566976 0.89 HSP90AB1 (0.79) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL4566979 0.89 HSP90AB1 (0.79) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL25602985 0.88 HSP90AB1 (0.78) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL419168 0.88 HSP90AB1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL421109 0.88 HSP90AB1 (0.78) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1854 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
US-20260137707-A1 METHODS OF MODULATING ATXN2 EXPRESSION UNIV OF UTAH RESEARCH FOUNDATION (US) 2026-05-21 US claimed
US-20260139320-A1 StarTrace: A Multiplex Drug Testing Platform for Personalized Medicine UNIV OF SOUTH CAROLINA (US) 2026-05-21 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-4729519-A1 CRYSTAL FORM OF ENPP1 INHIBITOR CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. (CN) 2026-04-22 EP claimed
US-20260102468-A1 COMPOSITIONS AND METHODS FOR MARCO INHIBITION AND IMPROVED DRUG DELIVERY UNIV TEXAS (US) 2026-04-16 US claimed
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms KARTOS THERAPEUTICS INC (US) 2026-04-09 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4695235-A1 NOVEL GSPT1 DEGRADER AND USE THEREOF Cyrus Therapeutics Inc. (KR) 2026-02-18 EP claimed
US-20260041673-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE BIOHAVEN THERAPEUTICS LTD (US) 2026-02-12 US claimed
EP-3373932-B1 CRYSTALLINE FORM OF A SUBSTITUTED QUINOLINE COMPOUND AND PHARMACEUTICAL COMPOSITIONS THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2022-03-30 EP claimed
WO-2022047008-A1 HSP90-BINDING CONJUGATES AND FORMULATIONS THEREOF TARVEDA THERAPEUTICS, INC. (US) 2022-03-03 WO claimed
US-20220054648-A1 ANTIBODY-DRUG CONJUGATES AND USES THEREOF IMMUNOMEDICS, INC. 2022-02-24 US claimed
US-11253606-B2 Combining anti-HLA-DR or anti-Trop-2 antibodies with microtubule inhibitors, PARP inhibitors, Bruton kinase inhibitors or phosphoinositide 3-kinase inhibitors significantly improves therapeutic outcome in cancer IMMUNOMEDICS, INC. (US) 2022-02-22 US claimed
EP-3954373-A1 NEOADJUVANT USE OF ANTIBODY-DRUG CONJUGATES Immunomedics, Inc. (US) 2022-02-16 EP claimed
CN-114040779-A Conjugates of cell binding molecules containing branched linkers and cytotoxic agents 杭州多禧生物科技有限公司 2022-02-11 CN claimed
CN-114040781-A Formulation of conjugate of TUBULYSIN derivative and cell binding molecule 杭州多禧生物科技有限公司 2022-02-11 CN claimed
CN-111214664-B Application of combination of USP2 and HSP90 inhibitor in inhibiting growth of ErbB2 positive breast cancer 大连医科大学 2022-02-11 CN claimed
US-11241500-B2 HSP90-targeting conjugates and formulations thereof TARVEDA THERAPEUTICS, INC. (US) 2022-02-08 US claimed
US-20220031853-A1 HSP90-TARGETING CONJUGATES AND FORMULATIONS THEREOF TVA (ABC), LLC 2022-02-03 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule CD4, TAP1, MCTS1 HSP90AB1 1068/4885HSP90AA1 1462/4885HSP90B1 1315/4885
US-20260097028-A1 Methods of Treating Myeloproliferative Neoplasms JAK2, TP53, CDKN1A HSP90AB1 233/4885HSP90AA1 291/4885HSP90B1 593/4885
US-20260137707-A1 METHODS OF MODULATING ATXN2 EXPRESSION ATXN2, ATXN2L, ATP6V1B2 HSP90AB1 38/4885HSP90AA1 60/4885HSP90B1 27/4885
US-20260041673-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE GFRA3, IL6ST, GFRA1 HSP90AB1 1512/4885HSP90AA1 2073/4885HSP90B1 3145/4885
US-20260139320-A1 StarTrace: A Multiplex Drug Testing Platform for Personalized Medicine PTH1R, SSTR4, MC4R HSP90AB1 3546/4885HSP90AA1 3615/4885HSP90B1 3365/4885
US-11241500-B2 HSP90-targeting conjugates and formulations thereof HSP90AB1, HSP90AA1, HSP90B1 HSP90AB1 1/4885HSP90AA1 2/4885HSP90B1 3/4885
US-20220031853-A1 HSP90-TARGETING CONJUGATES AND FORMULATIONS THEREOF HSP90AB1, HSP90AA1, HSP90B1 HSP90AB1 1/4885HSP90AA1 2/4885HSP90B1 3/4885
US-20260102468-A1 COMPOSITIONS AND METHODS FOR MARCO INHIBITION AND IMPROVED DRUG DELIVERY MSR1, TNFRSF9, TNFSF10 HSP90AB1 1286/4885HSP90AA1 1849/4885HSP90B1 1081/4885
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS DCLRE1A, CCR3, CCR8 HSP90AB1 2943/4885HSP90AA1 3328/4885HSP90B1 2973/4885
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF CHEK1, ATR, MRE11 HSP90AB1 2094/4885HSP90AA1 3097/4885HSP90B1 2166/4885
US-11253606-B2 Combining anti-HLA-DR or anti-Trop-2 antibodies with microtubule inhibitors, PARP inhibitors, Bruton kinase inhibitors or phosphoinositide 3-kinase inhibitors significantly improves therapeutic outcome in cancer PARP2, DOCK2, DYNLL2 HSP90AB1 286/4885HSP90AA1 437/4885HSP90B1 580/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.