SCHEMBL4199168

SCHEMBL4199168

CC(=O)Nc1ccc(N=Nc2ccc(C)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.77
SMN1; SMN2 Q16637 6/20 0.73
MAPT P10636 5/20 0.73
NPC1 O15118 5/20 0.73
RAB9A P51151 5/20 0.73
HPGD P15428 2/20 0.73
LMNA P02545 1/20 0.73
NFKB1 P19838 1/20 0.73
NFKB2 Q00653 1/20 0.73
RELA Q04206 1/20 0.73
THRB P10828 1/20 0.69
PKM P14618 2/20 0.61
MAPK1 P28482 1/20 0.58
STAT3 P40763 1/20 0.58
STAT1 P42224 1/20 0.58
HTT P42858 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 4/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18405965 1.00 TDP1 (0.77) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL12620630 1.00 TDP1 (0.77) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL11649000 0.92 MAPT (0.85) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL11648995 0.92 MAPT (0.85) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL19272225 0.92 MAPT (0.85) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL61417 0.88 TDP1 (1.00) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL19227683 0.86 SMN1; SMN2 (0.76) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL18409070 0.86 TDP1 (0.57) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL23259443 0.85 MAPT (1.00) TDP1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL1405623 0.85 MAPT (1.00) TDP1SMN1; SMN2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3621958-B1 PHOTOCHROMIC INDENO FUSED PHENANTHRENOPYRAN COMPOUNDS TRANSITIONS OPTICAL LTD (IE) 2024-07-10 EP disclosed
EP-3268375-B1 PHOTOCHROMIC THIENOCHROMENE COMPOUNDS TRANSITIONS OPTICAL INC (US) 2022-06-15 EP disclosed
EP-3071576-B9 PHOTOCHROMIC INDENO-FUSED RING PYRAN COMPOUNDS TRANSITIONS OPTICAL INC (US) 2021-12-22 EP disclosed
EP-3071576-B1 PHOTOCHROMIC INDENO-FUSED RING PYRAN COMPOUNDS TRANSITIONS OPTICAL INC (US) 2021-08-18 EP disclosed
EP-3071550-B1 METHOD OF PREPARING FUSED RING INDENO COMPOUNDS TRANSITIONS OPTICAL INC (US) 2019-03-13 EP disclosed
EP-1504918-B1 LAMINATE FOR PRINTING AND, PRINTING METHOD AND PRINTED MATTER USING THE SAME KIWA CHEMICAL IND CO LTD (JP) 2009-03-04 EP disclosed
EP-1415798-B1 LAMINATED BODY FOR PRINTING WITH TEMPORARY DISPLAY LAYER KIWA CHEMICAL IND CO LTD (JP) 2008-09-10 EP disclosed
EP-1504918-A1 LAMINATE FOR PRINTING AND, PRINTING METHOD AND PRINTED MATTER USING THE SAME Kiwa Chemical Industry Co., Ltd. (JP) 2005-02-09 EP disclosed
EP-1415798-A1 TEMPORARY DISPLAY LAYER CARRYING PRINTING LAMINATE Kiwa Chemical Industry Co., Ltd. (JP) 2004-05-06 EP disclosed