SCHEMBL4206605

SCHEMBL4206605

O=C(c1ccccc1)N1CCC(c2ccccc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.71
CA1 P00915 1/20 0.71
CA2 P00918 1/20 0.71
CA7 P43166 1/20 0.71
CA9 Q16790 1/20 0.71
CA14 Q9ULX7 1/20 0.71
SLC18A3 Q16572 1/20 0.68
ACHE P22303 1/20 0.67
HSD11B1 P28845 1/20 0.66
NPC1 O15118 1/20 0.66
RAB9A P51151 1/20 0.66
ATM Q13315 1/20 0.66
NAMPT P43490 1/20 0.64
EPHX1 P07099 1/20 0.61
L3MBTL3 Q96JM7 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
CCR5 P51681 1/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
HPGD P15428 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10720211 0.96 CA12 (0.76) CA12CA1CA2CA7CA9
SCHEMBL10720101 0.92 PARP14 (0.65) CA12CA1CA2CA7CA9
SCHEMBL12447384 0.90 RAB9A (0.81) CA12CA1CA2CA7CA9
SCHEMBL20006200 0.90 RAB9A (0.81) CA12CA1CA2CA7CA9
SCHEMBL21084408 0.89 LMNA (0.67) CA12CA1CA2CA7CA9
SCHEMBL27860960 0.89 CA12 (0.63) CA12CA1CA2CA7CA9
SCHEMBL95659 0.89 CA12 (0.67) CA12CA1CA2CA7CA9
SCHEMBL786718 0.89 NPC1 (0.84) CA12CA1CA2CA7CA9
SCHEMBL27629062 0.89 NPC1 (0.74) CA12CA1CA2CA7CA9
SCHEMBL13212972 0.89 CA12 (0.71) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501467-A4 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION BRISTOL MYERS SQUIBB CO (US) 2009-08-19 EP disclosed
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
EP-1501467-A2 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION Bristol-Myers Squibb Company (US) 2005-02-02 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed
WO-2003088908-A2 HETEROCYCLO INHIBITORS OF POTASSIUM CHANNEL FUNCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2003-10-30 WO disclosed