Losartan

Losartan

SCHEMBL42080

CCCCc1nc(Cl)c(CO)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1.[KH]

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 4/20 0.66
AGTR2 P50052 3/20 0.66
ABCC4 O15439 1/20 0.66
ABCB11 O95342 1/20 0.66
PDE3B Q13370 1/20 0.66
PDE3A Q14432 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Losartan SCHEMBL7420948 1.00 AGTR1 (0.66) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL4090171 1.00 AGTR1 (0.66) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL6684517 0.99 AGTR1 (0.65) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL6684460 0.99 AGTR1 (0.65) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL28493004 0.99 AGTR1 (0.65) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL60 0.99 AGTR1 (0.67) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL29383742 0.99 AGTR1 (0.67) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL6092394 0.99 AGTR1 (0.67) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL4726128 0.98 AGTR1 (0.66) AGTR1AGTR2ABCC4ABCB11PDE3B
Losartan SCHEMBL3216357 0.98 AGTR1 (0.66) AGTR1AGTR2ABCC4ABCB11PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8016 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12605365-B2 Losartan liquid formulations and methods of use SCIENTURE, LLC (US) 2026-04-21 US claimed
US-20260060963-A1 READY-TO-USE NON-AQUEOUS ORAL SOLUTION OF LOSARTAN LIQMEDS WORLDWIDE LIMITED (GB) 2026-03-05 US claimed
US-12496291-B1 Ready-to-use non-aqueous oral solution of losartan LIQMEDS WORLDWIDE LIMITED (GB) 2025-12-16 US claimed
EP-4638742-A1 COMPOSITIONS AND METHODS FOR INHIBITING EXPRESSION OF 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 13 (HSD17B13) Shanghai Argo Biopharmaceutical Co., Ltd. (CN) 2025-10-29 EP claimed
US-20250319070-A1 LOSARTAN LIQUID FORMULATIONS AND METHODS OF USE STREETERVILLE CAPITAL, LLC 2025-10-16 US claimed
WO-2025131019-A1 COMPOSITIONS AND METHODS FOR INHIBITING EXPRESSION OF INHIBIN SUBUNIT BETA E (INHBE) SHANGHAI ARGO BIOPHARMACEUTICAL CO., LTD. (CN) 2025-06-26 WO claimed
CN-120044164-A Method for detecting impurities in losartan potassium 珠海润都制药股份有限公司 2025-05-27 CN claimed
WO-2025090879-A1 PLURIPOTENT CELL DIFFERENTIATION AMGEN INC. (US) 2025-05-01 WO claimed
CN-119792218-A Stable metaxartan potassium tablet and preparation method thereof 江苏天士力帝益药业有限公司 2025-04-11 CN claimed
US-20250115584-A1 High-Purity Losartan Potassium and Preparation Method Therefor ZHEJIANG HUAHAI PHARMACEUTICAL CO., LTD. (CN) 2025-04-10 US claimed
WO-1998018787-A1 PROCESS FOR THE CRYSTALLIZATION OF LOSARTAN MERCK & CO., INC. (US) 1998-05-07 WO claimed
EP-0831911-A2 SPIRONOLACTONE AND ANGIOTENSIN II ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE G.D. SEARLE & CO. (US) 1998-04-01 EP claimed
EP-0831910-A1 EPOXY-STEROIDAL ALDOSTERONE ANTAGONIST AND ANGIOTENSIN II ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE G.D. SEARLE & CO. (US) 1998-04-01 EP claimed
EP-0733366-B1 Pharmaceutical compositions comprising angiotensin II receptor blocking imidazoles and diuretics DU PONT (US) 1998-04-01 EP claimed
WO-1997049392-A1 A COMPOSITION OF ENALAPRIL AND LOSARTAN MERCK & CO., INC. (US) 1997-12-31 WO claimed
WO-1996040255-A2 METHOD TO TREAT CARDIOFIBROSIS WITH A COMBINATION THERAPY OF AN ANGIOTENSIN II ANTAGONIST AND AN EPOXY-STEROIDAL ALDOSTERONE ANTAGONIST G.D. SEARLE & CO. (US) 1996-12-19 WO claimed
WO-1996040257-A1 EPOXY-STEROIDAL ALDOSTERONE ANTAGONIST AND ANGIOTENSIN II ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE G.D. SEARLE & CO. (US) 1996-12-19 WO claimed
WO-1996040258-A2 SPIRONOLACTONE AND ANGIOTENSIN II ANTAGONIST COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE G.D. SEARLE & CO. (US) 1996-12-19 WO claimed
WO-1996040256-A1 METHOD TO TREAT CARDIOFIBROSIS WITH A COMBINATION OF AN ANGIOTENSIN II ANTAGONIST AND SPIRONOLACTONE G.D. SEARLE & CO. (US) 1996-12-19 WO claimed
EP-0733366-A2 Pharmaceutical compositions comprising angiotensin II receptor blocking imidazoles and diuretics E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-09-25 EP claimed