SCHEMBL4209591

SCHEMBL4209591

CCc1n[nH]c(C(C)CCO)c1Oc1ccc(C#N)c(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.41
CYP19A1 P11511 1/20 0.34
PDE4B Q07343 4/20 0.33
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
PDE4A P27815 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
MAOB P27338 2/20 0.31
MAOA P21397 1/20 0.31
SLC5A1 P13866 1/20 0.31
SLC5A2 P31639 1/20 0.31
ACACB O00763 2/20 0.31
AR P10275 2/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4112181 0.78 KCNH2 (0.66) KCNH2CYP19A1PDE4BALDH1A1HPGD
SCHEMBL4112493 0.68 PGR (0.42) CYP19A1PDE4BALDH1A1HPGDMAOB
SCHEMBL4106178 0.68 KCNH2 (0.60) KCNH2CYP19A1AR
SCHEMBL4109289 0.66 KCNH2 (0.58) KCNH2AR
SCHEMBL509689 0.62 KCNH2 (0.79) KCNH2
SCHEMBL4581525 0.62 CYP19A1 (0.65) CYP19A1PDE4BALDH1A1HPGDMAOB
SCHEMBL29390509 0.62 CYP19A1 (0.65) CYP19A1PDE4BALDH1A1HPGDMAOB
SCHEMBL4141536 0.62 AR (0.51) CYP19A1PDE4BALDH1A1HPGDMAOB
SCHEMBL4109180 0.62 KCNH2 (0.75) KCNH2CYP19A1
SCHEMBL4104698 0.61 AR (0.43) CYP19A1PDE4BALDH1A1HPGDMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7482375-B2 Compounds useful in therapy PFIZER INC. (US) 2009-01-27 US disclosed