SCHEMBL4215088

SCHEMBL4215088

CCOC(=O)n1ncc2c(N)cccc21

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
ELANE P08246 11/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
F2 P00734 1/20 0.41
PLAU P00749 1/20 0.41
CDC25B P30305 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1855369 0.87 SCN9A (0.45) TP53ELANENPC1RAB9AHPGD
SCHEMBL1857119 0.85 NPC1 (0.45) TP53ELANENPC1RAB9AKMT2A
SCHEMBL21874382 0.84 HDAC1 (0.41) NPC1RAB9AKMT2AALDH1A1
SCHEMBL29510728 0.82 MAP2K4 (0.45) ELANENPC1RAB9AKMT2A
SCHEMBL2478647 0.82 MAP2K4 (0.45) ELANENPC1RAB9AKMT2A
SCHEMBL1863326 0.82 ELANE (0.46) ELANENPC1RAB9AHPGDKMT2A
SCHEMBL4787612 0.81 NPC1 (0.47) TP53ELANENPC1RAB9AHPGD
SCHEMBL3604733 0.80 CHEK1 (0.50) ELANENPC1RAB9AKMT2A
SCHEMBL13318330 0.79 DDB1 (0.41) ELANENPC1RAB9AHPGDKMT2A
SCHEMBL28337035 0.78 ELANE (0.50) ELANENPC1RAB9AHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2017265-A1 Fused compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor Abbott Laboratories (US) 2009-01-21 EP disclosed