SCHEMBL4222657

SCHEMBL4222657

N#Cc1ccc2c(c1)CCCC2(SCCO)c1c[nH]cn1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.40
CYP19A1 P11511 3/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
PGR P06401 1/20 0.31
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
PNMT P11086 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4437916 0.86 KDM1A (0.39) KDM1APGRDRD2DRD3PNMT
SCHEMBL733031 0.79 KDM1A (0.36) KDM1APGR
SCHEMBL731436 0.76 KDM1A (0.35) KDM1APGRDRD2DRD3
SCHEMBL733341 0.66 KDM1A (0.35) KDM1APGRDRD2DRD3
SCHEMBL4045639 0.64 KDM1A (0.34) KDM1APGRDRD2DRD3
SCHEMBL732031 0.63 KDM1A (0.46) KDM1ACYP19A1CYP11B1CYP11B2PGR
SCHEMBL17987977 0.58 KDM1A (1.00) KDM1ADRD2DRD3PNMT
SCHEMBL8746261 0.57 KDM1A (0.47) KDM1ACYP19A1CYP11B1CYP11B2PGR
SCHEMBL4226656 0.57 CYP19A1 (0.61) KDM1ACYP19A1CYP11B1CYP11B2DRD2
SCHEMBL4219622 0.57 CYP19A1 (0.61) KDM1ACYP19A1CYP11B1CYP11B2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010540-B1 SPIRO-IMIDAZO COMPOUNDS NOVARTIS AG (CH) 2012-12-05 EP disclosed
EP-2010540-A1 SPIRO-IMIDAZO COMPOUNDS Speedel Experimenta AG (CH) 2009-01-07 EP disclosed
WO-2007116098-A1 SPIRO-IMIDAZO COMPOUNDS SPEEDEL EXPERIMENTA AG (CH) 2007-10-18 WO disclosed