SCHEMBL733031

SCHEMBL733031

CCC(SC1(c2c[nH]cn2)CCCc2cc(C#N)ccc21)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.36
EP300 Q09472 1/20 0.32
CREBBP Q92793 1/20 0.32
PGR P06401 2/20 0.31
PTGES O14684 1/20 0.30
ALOX5 P09917 1/20 0.30
PPARG P37231 1/20 0.30
CXCR5 P32302 1/20 0.30
SLC22A12 Q96S37 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4437916 0.83 KDM1A (0.39) KDM1AEP300CREBBPPGRCXCR5
SCHEMBL731360 0.80 DRD2 (0.33) KDM1AEP300CREBBPPGRSYK
SCHEMBL4222657 0.79 KDM1A (0.40) KDM1APGR
SCHEMBL2917019 0.64 PTGES (0.35) PTGESALOX5PPARG
SCHEMBL4045639 0.62 KDM1A (0.34) KDM1AEP300CREBBPPGRCXCR5
SCHEMBL731083 0.61 DRD2 (0.33) KDM1AEP300CREBBPPGRSYK
SCHEMBL733341 0.61 KDM1A (0.35) KDM1APGRSYK
SCHEMBL17988227 0.60 KDM1A (0.66) KDM1APGRCXCR5
SCHEMBL4495832 0.59 KDM1A (0.42) KDM1AEP300CREBBPCXCR5
SCHEMBL4495829 0.59 KDM1A (0.42) KDM1AEP300CREBBPCXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138179-B2 Spiro-imidazo compounds NOVARTIS AG (CH) 2012-03-20 US disclosed