SCHEMBL4224922

SCHEMBL4224922

COC(=O)c1[nH]nc(C(=O)O)c1OCc1ccccc1.COC(=O)c1n[nH]c(C(=O)OC)c1OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
USP2 O75604 1/20 0.53
TSHR P16473 1/20 0.53
HSD17B10 Q99714 1/20 0.53
HPGD P15428 2/20 0.50
LMNA P02545 2/20 0.50
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4C Q9H3R0 1/20 0.44
KDM4E B2RXH2 2/20 0.44
STAT3 P40763 1/20 0.44
HIF1A Q16665 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.40
CCNB2 O95067 1/20 0.40
CCNE2 O96020 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4205180 0.97 ALDH1A1 (0.55) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL4205968 0.96 ALDH1A1 (0.56) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL13947735 0.92 HPGD (0.52) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL18655533 0.89 HPGD (0.51) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL4206891 0.85 NR4A2 (0.44) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL24906243 0.83 LMNA (0.53) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL23115819 0.83 ALDH1A1 (0.56) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL24906205 0.78 LMNA (0.48) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL4196581 0.78 ALDH1A1 (0.41) ALDH1A1USP2TSHRHSD17B10HPGD
SCHEMBL4196583 0.78 ALDH1A1 (0.41) ALDH1A1USP2TSHRHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758585-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2009-07-22 EP disclosed
EP-1758585-A2 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2007-03-07 EP disclosed
WO-2005120516-A2 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-12-22 WO disclosed