SCHEMBL4226593

SCHEMBL4226593

CC(=O)N(C)CCC1CN(Cc2ccc(F)cc2)C(=O)c2c(CC(=O)O)c(=O)n(C(C)C)c(=O)n21

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.34
ACHE P22303 2/20 0.34
AKR1B1 P15121 1/20 0.34
TP53 P04637 1/20 0.33
HMGCR P04035 1/20 0.32
KMT2A Q03164 2/20 0.32
ENPP2 Q13822 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PTGDR2 Q9Y5Y4 5/20 0.31
S1PR1 P21453 1/20 0.31
MEN1 O00255 1/20 0.31
PTGDR Q13258 1/20 0.30
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2891360 0.90 ACHE (0.34) HTTACHEAKR1B1TP53HMGCR
SCHEMBL2890889 0.86 ACHE (0.32) HTTACHETP53HMGCRKMT2A
Hydrochloric Acid SCHEMBL4224979 0.85 TP53 (0.36) HTTAKR1B1TP53HMGCRKMT2A
SCHEMBL2900634 0.81 ACHE (0.40) HTTACHEHMGCRKMT2A
SCHEMBL13085834 0.81 TP53 (0.35) HTTTP53HMGCRS1PR1GRM2
SCHEMBL2891857 0.80 TP53 (0.39) HTTAKR1B1TP53HMGCRKMT2A
SCHEMBL13094093 0.78 HTT (0.35) HTTTP53HMGCRKMT2AGRM2
SCHEMBL2892030 0.78 P2RX3 (0.33) HTTTP53HMGCRKMT2AL3MBTL1
SCHEMBL2899639 0.78 TP53 (0.36) HTTTP53HMGCRKMT2A
SCHEMBL2898698 0.77 KMT2A (0.39) HTTHMGCRKMT2AL3MBTL1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725102-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2009-04-29 EP disclosed
EP-1725102-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2006-11-29 EP disclosed
WO-2005092099-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-10-06 WO disclosed