SCHEMBL4227771

SCHEMBL4227771

N#Cc1ccc(NC(C(=O)NCC2CCCCC2)(c2ccccc2)C(F)(F)C(=O)OF)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNK O75909 2/20 0.40
CDK12 Q9NYV4 2/20 0.40
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CNR2 P34972 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
CETP P11597 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
OPRK1 P41145 1/20 0.36
AR P10275 1/20 0.36
CHRM4 P08173 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
USP30 Q70CQ3 1/20 0.35
CCR6 P51684 2/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237398 0.83 ABCB1 (0.42) CCNKCDK12CCNA2CDK2OPRM1
SCHEMBL4222280 0.82 CNR1 (0.36) CCNKCDK12CCNA2CDK2CNR2
SCHEMBL4228168 0.78 CCR6 (0.40) CHRM2CHRM1CHRM3CCR6
Trifluoroacetic Acid SCHEMBL4227766 0.72 MTTP (0.43) CCNKCDK12CCNA2CDK2OPRK1
SCHEMBL4232751 0.68
SCHEMBL22304147 0.68 TSHR (0.50) ALDH1A1OPRK1HDAC6EPHX1
SCHEMBL6820877 0.61 DPP4 (0.58) USP30HCRTR1
SCHEMBL1597146 0.61 DPP4 (0.58) USP30HCRTR1
SCHEMBL15739611 0.61 EGLN2 (0.51) USP30
SCHEMBL507198 0.61 CCR6 (0.55) CCNKCDK12CCNA2CDK2CCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2096104-A1 Organic diamines as mGluR7 modulators Novartis AG (CH) 2009-09-02 EP disclosed