SCHEMBL4229393

SCHEMBL4229393

CCCCN1CCC(Oc2ccc(C(=O)Nc3ccc(Oc4cc(F)c(NC(=O)NC(CC)CC)cc4F)cc3)cc2C)CC1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 7/20 0.38
ERBB2 P04626 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
BCL9 O00512 1/20 0.36
CTNNB1 P35222 1/20 0.36
FLT1 P17948 4/20 0.36
KDR P35968 4/20 0.36
TAS1R3 Q7RTX0 2/20 0.35
TAS1R1 Q7RTX1 2/20 0.35
WNT3A P56704 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687897 0.97 MCHR1 (0.36) MCHR1ERBB2HRH3MEN1POLB
SCHEMBL4233744 0.94 MAPT (0.39) MCHR1POLBMAPTTAS1R3TAS1R1
SCHEMBL4236667 0.93 TAS1R3 (0.40) MCHR1ERBB2HRH3MEN1POLB
SCHEMBL4233470 0.92 MCHR1 (0.40) MCHR1ERBB2HRH3MEN1POLB
SCHEMBL4232306 0.92 CCR3 (0.39) HRH3MEN1MAPTKMT2ATAS1R3
SCHEMBL4683749 0.91 LMNA (0.39) MCHR1ERBB2MEN1POLBMAPT
SCHEMBL4237351 0.90 LMNA (0.39) MCHR1ERBB2MEN1POLBMAPT
SCHEMBL4689324 0.90 CCR3 (0.44) MCHR1MEN1POLBMAPTKMT2A
SCHEMBL4236472 0.90 HRH3 (0.41) MCHR1HRH3MAPTBCL9CTNNB1
SCHEMBL4229188 0.90 MCHR1 (0.40) MCHR1ERBB2HRH3MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US claimed
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP claimed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO claimed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R MCHR1 47/4885ERBB2 348/4885HRH3 210/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.