SCHEMBL4229463

SCHEMBL4229463

OCCc1c[nH]c2cccc(Br)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.49
CYP2A6 P11509 1/20 0.47
HTR2A P28223 9/20 0.46
GPR84 Q9NQS5 3/20 0.46
HTR2B P41595 5/20 0.45
HTR1A P08908 2/20 0.45
DRD1 P21728 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR1E P28566 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
HTR5A P47898 1/20 0.45
HTR6 P50406 1/20 0.45
FFAR1 O14842 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25381397 0.86 CYP2A6 (0.50) HTR2CCYP2A6HTR2AGPR84HTR2B
SCHEMBL3478093 0.83 HTR2A (0.68) HTR2CCYP2A6HTR2AGPR84HTR2B
SCHEMBL18509280 0.81 GPR17 (0.55) HTR2CCYP2A6HTR2AHTR2BHTR1A
SCHEMBL3964357 0.81 GPR84 (0.71) HTR2CHTR2AGPR84HTR2BHTR1A
SCHEMBL19799203 0.81 HTR2C (0.73) HTR2CHTR2AGPR84HTR2BHTR1A
SCHEMBL29441748 0.81 HTR2C (0.73) HTR2CHTR2AGPR84HTR2BHTR1A
SCHEMBL15767915 0.79 HTR2A (0.73) HTR2CHTR2AGPR84HTR2BHTR1A
SCHEMBL4220443 0.79 GPR84 (0.69) HTR2CHTR2AGPR84HTR2BHTR1A
SCHEMBL30936114 0.79 HTR2A (0.68) HTR2CHTR2AHTR2BHTR1ADRD1
SCHEMBL19216922 0.79 CYP2A6 (0.54) HTR2CCYP2A6HTR2AGPR84HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006089-A2 A2 ADENOSINE RECEPTOR AGONISTS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2009-01-08 WO disclosed
US-5830911-A ANTIARTHRITIC AGENTS; ANTICARCINOGENIC AGENTS; ALZHEIMER'SDISEASE AMERICAN HOME PRODUCTS CORPORATION (US) 1998-11-03 US disclosed