SCHEMBL18509280

SCHEMBL18509280

O=C(O)CCc1c[nH]c2cccc(Br)c12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 3/20 0.55
GAA P10253 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
THRB P10828 1/20 0.50
DNMT1 P26358 1/20 0.50
RECQL P46063 1/20 0.50
CASP6 P55212 1/20 0.50
KMT2A Q03164 1/20 0.50
MCL1 Q07820 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.47
CYP2A6 P11509 1/20 0.46
HTR2C P28335 2/20 0.44
MTNR1A P48039 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562093 0.84 ALDH1A1 (0.69) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL15323836 0.83 GAA (0.72) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL16540351 0.82 GPR17 (0.69) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL20935015 0.82 GPR17 (0.54) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL15141741 0.82 HTR2A (0.65) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL15142475 0.82 GPR84 (0.61) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL31036403 0.82 GPR84 (0.61) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL4229463 0.81 HTR2C (0.49) GAAKDM4EMEN1ALDH1A1POLB
SCHEMBL7917193 0.81 GPR17 (0.56) GPR17GAAKDM4EMEN1ALDH1A1
SCHEMBL18509792 0.79 PTGER1 (0.51) GPR17GAAKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081456-A1 HIGHLY ACTIVE SELF-SUFFICIENT NITRATION BIOCATALYSTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2018-05-03 WO disclosed
WO-2016134145-A9 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2017-02-16 WO disclosed