SCHEMBL4230615

SCHEMBL4230615

COc1ccc(CC(=O)NC2CCN(CCCN3C=COC(C4=C(Cl)C=CC(=O)C4)=C3)CC2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 5/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
SIGMAR1 Q99720 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.44
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 1/20 0.41
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
CHRM2 P08172 1/20 0.39
ADRA2A P08913 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2B P18089 1/20 0.39
CHRM3 P20309 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4235669 0.91 CHRM1 (0.55) CHRM1CHRM4CHRM5SIGMAR1SMN1; SMN2
SCHEMBL4226945 0.78 CHRM1 (0.45) CHRM1CHRM4CHRM5CHRM2DRD2
SCHEMBL4051360 0.78 SIGMAR1 (0.47) CHRM1CHRM4CHRM5SIGMAR1CHRM2
SCHEMBL4231625 0.77 CHRM1 (0.53) CHRM1CHRM4CHRM5SIGMAR1
SCHEMBL4049616 0.76 SIGMAR1 (0.49) CHRM1CHRM4CHRM5SIGMAR1CHRM2
SCHEMBL1554091 0.73 CHRM1 (0.49) CHRM1CHRM4CHRM5SIGMAR1CHRM2
SCHEMBL4230607 0.69 CHRM1 (0.65) CHRM1CHRM4CHRM5SIGMAR1SMN1; SMN2
SCHEMBL4055943 0.68 CHRM1 (1.00) CHRM1CHRM4CHRM5SIGMAR1SMN1; SMN2
SCHEMBL2406403 0.67 SIGMAR1 (0.70) SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL4049143 0.67 CHRM1 (0.35) CHRM1CHRM4CHRM5ALDH1A1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009106534-A1 NOVEL HETEROCYCLIC CARBOXAMIDES AS M1 AGONISTS H. LUNDBECK A/S (DK) 2009-09-03 WO claimed
WO-2009106534-A1 NOVEL HETEROCYCLIC CARBOXAMIDES AS M1 AGONISTS H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed