SCHEMBL4233418

SCHEMBL4233418

CCCCN1CCC(Oc2ccc(C(=O)Nc3ccc(Oc4ccc(NC(=O)NC(CC)CC)cc4Cl)cc3F)cc2C)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.38
UBE2M P61081 2/20 0.37
DCUN1D1 Q96GG9 2/20 0.37
KDR P35968 4/20 0.37
FGFR1 P11362 1/20 0.37
CHRM1 P11229 1/20 0.37
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC2A1 P11166 1/20 0.36
UTS2R Q9UKP6 1/20 0.36
FLT1 P17948 2/20 0.36
FLT4 P35916 1/20 0.36
BRAF P15056 1/20 0.36
ERBB2 P04626 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4226808 0.93 CCR3 (0.40) MCHR1UBE2MDCUN1D1KDRFGFR1
SCHEMBL4229188 0.93 MCHR1 (0.40) MCHR1KDRMEN1POLBMAPT
SCHEMBL4238135 0.92 SMN1; SMN2 (0.41) MCHR1KDRFGFR1MEN1POLB
SCHEMBL4235427 0.92 TAS1R3 (0.40) MCHR1KDRMEN1POLBMAPT
SCHEMBL4238014 0.91 PKM (0.40) MCHR1KDRFLT1ERBB2
SCHEMBL4686866 0.90 CCR3 (0.44) MCHR1KDRMEN1POLBMAPT
SCHEMBL4233470 0.90 MCHR1 (0.40) MCHR1KDRMEN1POLBMAPT
SCHEMBL4228632 0.87 MCHR1 (0.39) MCHR1KDRFGFR1MEN1POLB
SCHEMBL4238724 0.85 MCHR1 (0.37) MCHR1KDRFGFR1MEN1POLB
SCHEMBL4240643 0.85 PDE4D (0.42) MCHR1KDRPOLBMAPTFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US claimed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP disclosed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R MCHR1 47/4885UBE2M 4675/4885DCUN1D1 4362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.