SCHEMBL42349

SCHEMBL42349

N#Cc1ccc(N)cn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28038567 0.98 CHEK1 (0.38)
SCHEMBL17539134 0.85 ALOX5AP (0.42)
SCHEMBL17502178 0.83 ALDH1A1 (0.50)
SCHEMBL30859509 0.82 P4HTM (0.44)
SCHEMBL3413808 0.80 ALDH1A1 (0.52)
SCHEMBL17539186 0.78 CHEK1 (0.53)
SCHEMBL17539185 0.78 CYP3A4 (0.50)
SCHEMBL18419348 0.76
SCHEMBL7085448 0.74 PDE10A (0.42)
SCHEMBL7642979 0.74 PDE10A (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1195 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115028642-B Diaryl dihydrofuro [3,4-d ] pyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2024-07-12 CN claimed
CN-108976325-B Amidoxime pyridine chelate resin and preparation method thereof 海南师范大学 2020-07-31 CN claimed
CN-108976325-A A kind of amidoxime group pyridine chelating resin and preparation method thereof 海南师范大学 2018-12-11 CN claimed
CN-105175453-B A kind of manganese complex is prepared and its synthetic method 合肥工业大学 2017-09-26 CN claimed
CN-105669710-B A kind of preparation of copper complex crystal and its synthetic method 合肥祥晨化工有限公司 2017-08-29 CN claimed
CN-105669772-A Preparation and synthesis method of nickel complex 合肥祥晨化工有限公司 2016-06-15 CN claimed
CN-105669710-A Preparation method and synthetic method for copper complex crystal 合肥祥晨化工有限公司 2016-06-15 CN claimed
CN-105175453-A Manganese complex preparation and synthesis method UNIV HEFEI TECHNOLOGY 2015-12-23 CN claimed
EP-2507243-B1 SPIROINDOLINONE PYRROLIDINES HOFFMANN LA ROCHE (CH) 2015-06-10 EP claimed
EP-2507243-A1 SPIROINDOLINONE PYRROLIDINES F. Hoffmann-La Roche AG (CH) 2012-10-10 EP claimed
JP-2006500348-A 2006-01-05 JP claimed
US-20050197349-A1 Pyrrolo[2,3-D]pyrimidine compounds PFIZER INC. 2005-09-08 US claimed
WO-2005066155-A1 5-FLUORO-, CHLORO- AND CYANO-PYRIDIN-2-YL-TETRAZOLES AS LIGANDS OF THE METABOTROPIC GLUTAMATE RECEPTOR-5 ASTRAZENECA AB (SE) 2005-07-21 WO claimed
EP-1534685-A1 1H-INDAZOLE-3-CARBOXAMIDE COMPOUNDS AS CYCLIN DEPENDENT KINASES (CDK) INHIBITORS Astex Technology Limited (GB) 2005-06-01 EP claimed
US-6696567-B2 INHIBITION OF PROTEIN KINASES OR JANUS KINASE 3; TREATING OR PREVENTING ORGAN TRANSPLANT REJECTION, XENO TRANSPLATION, LUPUS, MULTIPLE SCLEROSIS, RHEUMATOID ARTHRITIS, PSORIASIS, TYPE I DIABETES OR VARIOUS DISEASE COMPLICATIONS PFIZER INC. 2004-02-24 US claimed
WO-2004014864-A1 1H-INDAZOLE-3-CARBOXAMIDE COMPOUNDS AS CYCLIN DEPENDENT KINASES (CDK) INHIBITORS ASTEX TECHNOLOGY LIMITED (GB) 2004-02-19 WO claimed
US-20030220353-A1 Pyrrolo[2,3-d]pyrimidine compounds PFIZER INC. 2003-11-27 US claimed
EP-1294724-A1 PYRROLO[2,3-D]PYRIMIDINE COMPOUNDS AS IMMUNOSUPPRESSIVE AGENTS Pfizer Products Inc. (US) 2003-03-26 EP claimed
US-20020068746-A1 Pyrrolo[2,3-d]pyrimidine compounds PFIZER INC. 2002-06-06 US claimed
WO-2002000661-A1 PYRROLO[2,3-d]PYRIMIDINE COMPOUNDS AS IMMUNOSUPPRESSIVE AGENTS PFIZER PRODUCTS INC. (US) 2002-01-03 WO claimed