SCHEMBL4237642

SCHEMBL4237642

CN(C)/C=C/C(=O)c1cccc(S(=O)(=O)NCCN(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
MAPT P10636 4/20 0.51
GAA P10253 3/20 0.51
HTT P42858 3/20 0.51
HPGD P15428 1/20 0.51
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
RECQL P46063 1/20 0.48
PKM P14618 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
AKR1C3 P42330 4/20 0.46
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MEP1B Q16820 1/20 0.45
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237644 1.00 ALDH1A1 (0.51) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL4056415 0.93 CYP2C19 (0.50) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL4056421 0.93 CYP2C19 (0.50) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL4059271 0.87 CYP2C19 (0.54) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL4059267 0.87 CYP2C19 (0.54) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL4052733 0.83 MAPT (0.57) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL4059272 0.83 ALDH1A1 (0.63) ALDH1A1CYP2C19SMN1; SMN2PKMMAPK1
SCHEMBL4052735 0.83 MAPT (0.57) ALDH1A1MAPTGAAHTTHPGD
SCHEMBL26731607 0.83 CYP2C19 (0.70) ALDH1A1HTTCYP2C19PKMMAPK1
SCHEMBL2850679 0.82 CYP2C19 (0.53) ALDH1A1HTTCYP2C19PKMMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111260-A1 PHENYLSULFONAMIDE-SUBSTITUTED, PYRAZOLO[1, 5-A]PYRIMIDINES, METHODS FOR PREPARATION AND USES THEREOF WYETH (US) 2009-09-11 WO disclosed