SCHEMBL4239254

SCHEMBL4239254

CCOc1cc(CN2CCC(N(c3ncccn3)N(c3ncccn3)C3CCNCC3)CC2)cc(OCC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
SSTR5 P35346 2/20 0.38
MCHR1 Q99705 1/20 0.38
HRH1 P35367 1/20 0.38
HTR2B P41595 1/20 0.38
ALDH1A1 P00352 4/20 0.37
KCNH2 Q12809 1/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
GMNN O75496 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
PMP22 Q01453 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4234624 0.87 ALDH1A1 (0.45) SLC6A2SLC6A4SLC6A3SSTR5ALDH1A1
SCHEMBL4225162 0.87 CYP19A1 (0.39) SLC6A2SLC6A4SSTR5HRH1HTR2B
SCHEMBL4232088 0.86 SSTR5 (0.44) SSTR5HRH1HTR2BALDH1A1KCNH2
SCHEMBL4232885 0.86 SSTR5 (0.46) SSTR5HRH1ALDH1A1KCNH2DRD2
SCHEMBL4236623 0.86 SSTR5 (0.41) SLC6A2SLC6A4SLC6A3SSTR5ALDH1A1
SCHEMBL4232220 0.86 SSTR5 (0.46) SSTR5HRH1ALDH1A1KCNH2DRD2
Hydrochloric Acid SCHEMBL4232793 0.84 PAX8 (0.39) SSTR5MCHR1KCNH2DRD2DRD4
SCHEMBL4233908 0.83 SSTR5 (0.44) SSTR5HRH1HTR2BALDH1A1KCNH2
SCHEMBL4234997 0.83 MAPT (0.36) SLC6A2SLC6A4SLC6A3SSTR5ALDH1A1
SCHEMBL4954333 0.82 SSTR5 (0.42) SSTR5MCHR1HRH1HTR2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-B1 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-07-01 EP disclosed