SCHEMBL4240205

SCHEMBL4240205

CN1C2CCCC1C(Oc1ccc(C(=O)O)cc1)C2

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 5/20 0.59
CHRM4 P08173 5/20 0.59
CHRM1 P11229 5/20 0.59
CHRM3 P20309 5/20 0.59
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4236286 0.78 HRH3 (0.51) CHRM2CHRM4CHRM1CHRM3
SCHEMBL13699322 0.77 EPHX2 (0.43) EPHX2
SCHEMBL4236560 0.77 SLC6A2 (0.67) CHRM2CHRM4CHRM1CHRM3EPHX2
SCHEMBL8437114 0.74 ALDH1A1 (0.56) EPHX2
SCHEMBL27917122 0.74 CHRM2 (1.00) CHRM2CHRM4CHRM1CHRM3
SCHEMBL11755572 0.71 PARP10 (0.71) EPHX2
SCHEMBL27516126 0.71 ALDH1A1 (0.49) EPHX2
SCHEMBL16701853 0.70 HRH3 (0.61) EPHX2
SCHEMBL4236506 0.70 ALDH1A1 (0.55) EPHX2
SCHEMBL13699096 0.70 ALDH1A1 (0.55) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP disclosed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R CHRM2 120/4885CHRM4 149/4885CHRM1 122/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.