SCHEMBL4240239

SCHEMBL4240239

CCCn1cc(-c2csc(Nc3ccccn3)n2)c(C(F)(F)F)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 17/20 0.50
RAB9A P51151 16/20 0.50
MEN1 O00255 13/20 0.50
KMT2A Q03164 13/20 0.50
MECP2 P51608 1/20 0.49
KCNN1 Q92952 1/20 0.49
KCNN2 Q9H2S1 1/20 0.49
MBD2 Q9UBB5 1/20 0.49
KCNN3 Q9UGI6 1/20 0.49
GRM4 Q14833 2/20 0.48
MAPT P10636 6/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
NFKB1 P19838 3/20 0.47
NFKB2 Q00653 3/20 0.47
RELA Q04206 3/20 0.47
TP53 P04637 3/20 0.47
LMNA P02545 3/20 0.47
MAPK1 P28482 3/20 0.47
GAA P10253 3/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4058319 0.86 NPC1 (0.55) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL3354574 0.83 NPC1 (0.56) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL4236252 0.82 ACHE (0.36) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL4241589 0.76 NPC1 (0.59) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL370409 0.74 GRM4 (0.57) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL4237850 0.72 NPC1 (0.56) NPC1RAB9AMEN1KMT2AGRM4
SCHEMBL4061311 0.70 MEN1 (0.57) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL4064704 0.70 NPC1 (0.62) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL4241658 0.69 NPC1 (0.58) NPC1RAB9AMEN1KMT2AMECP2
SCHEMBL3354435 0.69 NPC1 (0.58) NPC1RAB9AMEN1KMT2AMECP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO claimed