SCHEMBL4236252

SCHEMBL4236252

CCCn1cc(-c2nsc(Nc3ccccn3)n2)c(C(F)(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
KDR P35968 4/20 0.33
LRRK2 Q5S007 1/20 0.33
NPC1 O15118 7/20 0.32
RAB9A P51151 7/20 0.32
MEN1 O00255 6/20 0.32
KMT2A Q03164 6/20 0.32
MECP2 P51608 1/20 0.32
KCNN1 Q92952 1/20 0.32
KCNN2 Q9H2S1 1/20 0.32
MBD2 Q9UBB5 1/20 0.32
KCNN3 Q9UGI6 1/20 0.32
PDE5A O76074 1/20 0.32
MPL P40238 2/20 0.32
GRM4 Q14833 1/20 0.31
LMNA P02545 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPK10 P53779 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4240239 0.82 NPC1 (0.50) TRPV4NPC1RAB9AMEN1KMT2A
SCHEMBL4237345 0.77 KDR (0.40) ACHETRPV4KDRNPC1RAB9A
SCHEMBL4241119 0.75 ACHE (0.41) ACHETRPV4LRRK2MPL
SCHEMBL3357491 0.74 GRM4 (0.38) TRPV4KDRNPC1RAB9AMEN1
SCHEMBL4239555 0.70 TRPV4 (0.41) ACHETRPV4KDRNPC1RAB9A
SCHEMBL3356349 0.70 MEN1 (0.41) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL4235797 0.70 KDR (0.40) KDRNPC1RAB9AMEN1KMT2A
SCHEMBL4058319 0.69 NPC1 (0.55) TRPV4NPC1RAB9AMEN1KMT2A
SCHEMBL3357298 0.69 MEN1 (0.43) ACHENPC1RAB9AMEN1KMT2A
SCHEMBL15688006 0.68 MECP2 (0.46) KDRNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO disclosed