SCHEMBL4240823

SCHEMBL4240823

CCCCN1CCC(Oc2ccc(C#N)cc2)C(F)C1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.57
HRH2 P25021 9/20 0.52
HRH1 P35367 9/20 0.52
SIGMAR1 Q99720 2/20 0.49
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237843 0.84 HRH3 (0.72) HRH3HRH2HRH1SIGMAR1
SCHEMBL4240622 0.81 HRH2 (0.47) HRH3HRH2HRH1
SCHEMBL4237104 0.81 HRH3 (0.85) HRH3HRH2HRH1SIGMAR1MEN1
SCHEMBL4237090 0.77 HRH3 (0.46) HRH3HRH2HRH1SIGMAR1MEN1
SCHEMBL5206619 0.73 HRH3 (1.00) HRH3HRH2HRH1SIGMAR1
SCHEMBL7745171 0.72 MEN1 (0.51) HRH3HRH2HRH1SIGMAR1MEN1
SCHEMBL7745176 0.72 MEN1 (0.51) HRH3HRH2HRH1SIGMAR1MEN1
SCHEMBL7745173 0.72 MEN1 (0.51) HRH3HRH2HRH1SIGMAR1MEN1
SCHEMBL1715421 0.71 HRH3 (0.93) HRH3HRH2HRH1MEN1
SCHEMBL5208517 0.71 HRH3 (1.00) HRH3HRH2HRH1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R HRH3 210/4885HRH2 162/4885HRH1 217/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.