SCHEMBL4240850

SCHEMBL4240850

CCC(CC)NC(=O)Nc1ccc(Oc2ccc(N)cc2)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.53
PNLIP P16233 11/20 0.52
GCGR P47871 1/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
PARG Q86W56 1/20 0.44
STK39 Q9UEW8 1/20 0.44
F7 P08709 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4238208 0.89 PKM (0.53) PKMPNLIPGCGRMAPTNPSR1
SCHEMBL4236606 0.89 PKM (0.56) PKMPNLIPGCGRMAPTNPSR1
SCHEMBL4228260 0.87 PKM (0.54) PKMMAPTTAS1R3TAS1R1STK39
SCHEMBL4238927 0.87 PKM (0.54) PKMPNLIPMAPTTAS1R3TAS1R1
SCHEMBL5181890 0.87 PNLIP (0.55) PNLIPGCGRMAPTNPSR1PARG
SCHEMBL4228811 0.86 PKM (0.60) PKMMAPTNPSR1TAS1R3TAS1R1
SCHEMBL4229305 0.86 PKM (0.60) PKMMAPTTAS1R3TAS1R1
SCHEMBL4236991 0.86 PKM (0.53) PKMPNLIPMAPTTAS1R3TAS1R1
SCHEMBL4231850 0.86 PKM (0.48) PKMPNLIPGCGRMAPTNPSR1
Ammonia Solution, Strong SCHEMBL4235457 0.85 PKM (0.58) PKMMAPTNPSR1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP disclosed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R PKM 1734/4885PNLIP 1855/4885GCGR 66/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.