SCHEMBL4242685

SCHEMBL4242685

N[C@@H](Cc1ccc(CCCc2ccc3c(n2)NCCC3)cc1)C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.64
ITGA5 P08648 1/20 0.64
ITGAV P06756 19/20 0.55
ITGB3 P05106 17/20 0.55
ITGB5 P18084 3/20 0.55
ITGA2B P08514 4/20 0.53
ITGB6 P18564 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6224024 0.89 ITGAV (0.65) ITGB1ITGA5ITGAVITGB3ITGB5
SCHEMBL4245742 0.88 ITGB1 (0.58) ITGB1ITGA5ITGAVITGB3ITGB5
SCHEMBL4247583 0.85 ITGAV (0.52) ITGB1ITGA5ITGAVITGB3ITGB5
SCHEMBL4786884 0.85 ITGB3 (0.71) ITGB1ITGA5ITGAVITGB3ITGB5
SCHEMBL21853029 0.84 ITGAV (0.66) ITGAVITGB3ITGB6
SCHEMBL19953649 0.84 ITGAV (0.66) ITGAVITGB3ITGB6
SCHEMBL6421086 0.84 ITGAV (0.66) ITGAVITGB3ITGB6
Hydrochloric Acid SCHEMBL21853132 0.83 ITGAV (0.64) ITGAVITGB3ITGB6
Hydrochloric Acid SCHEMBL21853130 0.83 ITGAV (0.64) ITGAVITGB3ITGB6
Hydrochloric Acid SCHEMBL21853057 0.83 ITGAV (0.64) ITGAVITGB3ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049490-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL]-L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS Astra Zeneca AB (SE) 2009-04-22 EP disclosed
WO-2007141473-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL] -L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS ASTRAZENECA AB (SE) 2007-12-13 WO disclosed