Benzamide

Benzamide

SCHEMBL424272

COc1cc2c(-c3ccc(-c4ccccc4)cc3)ccc(N(C)C(=O)c3c(Br)ccc4c3OCO4)c2cc1OC.NC(=O)c1ccccc1

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.37
TARBP2 Q15633 1/20 0.36
RORC P51449 2/20 0.36
CHEK1 O14757 1/20 0.35
CHEK2 O96017 1/20 0.35
TP53 P04637 1/20 0.34
CYP1A2 P05177 2/20 0.32
HPGD P15428 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
EDNRB P24530 2/20 0.32
EDNRA P25101 2/20 0.32
CHUK O15111 1/20 0.32
INSR P06213 1/20 0.32
MAPK8 P45983 1/20 0.32
CAMKK2 Q96RR4 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
PDE2A O00408 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL419335 0.94 NPSR1 (0.38) NPSR1TARBP2TP53CYP1A2HPGD
SCHEMBL10132591 0.80 NPSR1 (0.42) NPSR1TARBP2TP53CYP1A2CYP2D6
SCHEMBL10132602 0.78 NPSR1 (0.43) NPSR1TARBP2TP53CYP1A2HPGD
SCHEMBL13283977 0.78 HTT (0.40) NPSR1RORCCYP1A2HPGDCYP2D6
SCHEMBL10132869 0.77 CYP19A1 (0.36) NPSR1HPGDEDNRAHTR2AHTR2C
SCHEMBL420470 0.77 MAPT (0.44) NPSR1TP53CYP1A2HPGDCYP1B1
SCHEMBL10132857 0.77 NPSR1 (0.38) NPSR1TP53PDE4APDE4BPDE4C
SCHEMBL10162945 0.76 HTT (0.41) NPSR1CYP1A2HPGDCYP2D6CYP2C19
SCHEMBL10132737 0.74 HTT (0.38) NPSR1RORCCYP1A2HPGDCYP2D6
SCHEMBL10132636 0.74 NPSR1 (0.42) NPSR1TARBP2TP53CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8741917-B2 Benzo [C] phenanthridines as antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-06-03 US disclosed
US-20120022061-A1 BENZO [C] PHENANTHRIDINES AS ANTIMICROBIAL AGENTS RUGTERS, THE STATE UNIVERSITY OF NEW JERSEY 2012-01-26 US disclosed
EP-2387564-A1 BENZO ÝC¨PHENANTHRIDINES AS ANTIMICROBIAL AGENTS Rutgers, The State University of New Jersey (US) 2011-11-23 EP disclosed
US-8037884-B2 Modular system for patient positioning during medical procedures ALLEN MEDICAL SYSTEMS, INC. (US) 2011-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120022061-A1 BENZO [C] PHENANTHRIDINES AS ANTIMICROBIAL AGENTS CCNT1, XPO4, XDH NPSR1 1352/4885TARBP2 3659/4885RORC 1630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.