SCHEMBL4243906

SCHEMBL4243906

CN(C)C(=O)N[C@@H](C[C@@H](O)CN(Cc1cncs1)C(=O)O)C(Cc1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 20/20 0.41
CYP2D6 P10635 3/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
MEN1 O00255 1/20 0.39
SLC22A2 O15244 1/20 0.39
SLC22A1 O15245 1/20 0.39
ABCC3 O15438 1/20 0.39
ABCC4 O15439 1/20 0.39
MLNR O43193 1/20 0.39
NR1I2 O75469 1/20 0.39
SLCO2B1 O94956 1/20 0.39
ABCB11 O95342 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PGR P06401 1/20 0.39
ABCB1 P08183 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943724 0.83 CYP3A4 (0.39) CYP3A4CYP2D6CYP2C19CYP1A2MEN1
SCHEMBL4248588 0.78 CYP3A4 (0.49) CYP3A4CYP2D6CYP2C19MEN1SLC22A2
SCHEMBL892851 0.72 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C19CYP1A2MEN1
SCHEMBL892849 0.72 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C19CYP1A2MEN1
SCHEMBL9943723 0.69 CYP3A4 (0.44) CYP3A4CYP2D6CYP2C19MEN1SLC22A2
SCHEMBL4245252 0.68 CYP3A4 (0.52) CYP3A4CYP2D6
SCHEMBL4251351 0.67 CYP3A4 (0.44) CYP3A4CYP2D6CYP2C19MEN1SLC22A2
SCHEMBL893249 0.67 CYP3A4 (0.65) CYP3A4CYP2D6CYP2C19CYP1A2MEN1
SCHEMBL9943656 0.67 CYP3A4 (0.67) CYP3A4
SCHEMBL15967935 0.67 ACACB (0.39) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed