SCHEMBL4245155

SCHEMBL4245155

NS(=O)(=O)CCc1ncccn1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.41
APLNR P35414 1/20 0.38
NAAA Q02083 1/20 0.36
AURKA O14965 1/20 0.36
DHFR P00374 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
CA2 P00918 6/20 0.34
CA1 P00915 2/20 0.33
CA9 Q16790 2/20 0.33
MAPK1 P28482 1/20 0.33
CA5A P35218 1/20 0.32
ENPP1 P22413 1/20 0.32
P2RX7 Q99572 1/20 0.31
PRMT1 Q99873 1/20 0.31
HSP90AA1 P07900 1/20 0.31
FTO Q9C0B1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26097655 0.79 APLNR (0.39) APLNRNAAAAURKADHFRLMNA
SCHEMBL19550276 0.77 APLNR (0.47) RECQLAPLNRLMNACA2CA1
SCHEMBL18247004 0.77 APLNR (0.67) RECQLAPLNRCA2CA1CA9
SCHEMBL18247184 0.77 APLNR (0.43) RECQLAPLNRCA2CA1CA9
SCHEMBL1154520 0.76 CA1 (0.44) AURKADHFRLMNATSHRCA2
SCHEMBL4184428 0.75 HRH1 (0.57) LMNACA2CA1PRMT1
Potassium SCHEMBL4063307 0.74 HRH1 (0.55) LMNACA2CA1PRMT1
SCHEMBL4063300 0.74 HRH1 (0.55) LMNACA2CA1PRMT1
SCHEMBL29170700 0.70 NAAA (0.42) APLNRNAAALMNA
Ethanesulfonic Acid Amide SCHEMBL16569730 0.70 COMT (0.38) AURKADHFRLMNATSHRCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049494-A2 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP claimed
WO-2008008310-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2008-01-17 WO claimed