SCHEMBL4245771

SCHEMBL4245771

CS(=O)(=O)Nc1ccc(C(N)=O)cc1.O=C(O)N1CCC(Oc2ccc(Cl)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.45
EPHX2 P34913 7/20 0.45
HRH1 P35367 1/20 0.44
CCR3 P51677 1/20 0.44
FAAH O00519 1/20 0.44
GRIN2D O15399 2/20 0.43
GRIN3B O60391 2/20 0.43
GRIN1 Q05586 2/20 0.43
GRIN2A Q12879 2/20 0.43
GRIN2B Q13224 2/20 0.43
GRIN2C Q14957 2/20 0.43
GRIN3A Q8TCU5 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2J2 P51589 1/20 0.43
NPY2R P49146 1/20 0.43
FPR2 P25090 2/20 0.40
PROKR1 Q8TCW9 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4244665 0.86 EPHX2 (0.50) PARP10EPHX2FAAHGRIN2DGRIN3B
SCHEMBL4244649 0.83 PARP10 (0.53) PARP10EPHX2FAAHGRIN2DGRIN3B
SCHEMBL27900126 0.81 PARP10 (0.67) PARP10EPHX2KMT2ACHEK2
SCHEMBL1256120 0.79 EPHX2 (0.60) EPHX2HRH1CCR3GRIN2DGRIN3B
SCHEMBL1805653 0.78 PARP10 (0.58) PARP10HRH3MEN1KMT2A
SCHEMBL4244552 0.77 PARP10 (0.57) PARP10EPHX2CYP2C9CYP2J2NPC1
SCHEMBL1808122 0.75 HRH3 (0.55) PARP10HRH3MEN1KMT2A
SCHEMBL1807050 0.75 HRH3 (0.52) EPHX2HRH1CCR3HRH3KMT2A
SCHEMBL4244729 0.74 GAA (0.56) FAAH
SCHEMBL1810548 0.74 HRH3 (0.50) EPHX2HRH1CCR3HRH3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170901-A1 Benzoyl Urea Derivatives RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170901-A1 Benzoyl Urea Derivatives OPRM1, GRIN2C, GRIN3A PARP10 3694/4885EPHX2 1860/4885HRH1 42/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.