SCHEMBL4246586

SCHEMBL4246586

CC1=C([C@H]2CCC[C@@H](c3ncccc3C)N2Cc2ccc(C#N)cc2CO)NCC=C1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 4/20 0.34
PARP1 P09874 1/20 0.32
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
PDE4A P27815 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
P2RX7 Q99572 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2472931 0.89 CXCR4 (0.40) CXCR4DDB1CRBNPDE4AKDM4E
SCHEMBL2473381 0.89 CXCR4 (0.40) CXCR4DDB1CRBNPDE4AKDM4E
SCHEMBL11904060 0.88 CXCR4 (0.33) CXCR4P2RX7
SCHEMBL15387270 0.82 CXCR4 (0.33) CXCR4
SCHEMBL2472797 0.79 CXCR4 (0.34) CXCR4KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL2477025 0.78 P2RX7 (0.38) DDB1CRBNALDH1A1P2RX7CYP11B2
SCHEMBL2476959 0.78 CXCR4 (0.35) CXCR4
SCHEMBL2470276 0.76 AR (0.37) KDM4EALDH1A1CYP1A2CYP3A4GAA
SCHEMBL2476471 0.76 AR (0.37) KDM4EALDH1A1CYP1A2CYP3A4GAA
SCHEMBL8301709 0.76 CXCR4 (0.40) CXCR4PARP1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550484-B2 Chemokine receptor binding heterocyclic compounds with enhanced efficacy GENZYME CORPORATION (US) 2009-06-23 US disclosed