SCHEMBL4246687

SCHEMBL4246687

CC[Al](Cl)Oc1c(C(C)(C)C)cc(C(C)(C)C)cc1C(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
RXRA P19793 7/20 0.32
PPARG P37231 7/20 0.32
RARG P13631 2/20 0.32
NR5A2 O00482 1/20 0.31
NR5A1 Q13285 1/20 0.31
RARA P10276 2/20 0.30
RARB P10826 2/20 0.30
RXRB P28702 2/20 0.30
RXRG P48443 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8859882 0.86 SMN1; SMN2 (0.39) CYP3A4CYP2C9CYP2C19
SCHEMBL8859887 0.84 PTGDR2 (0.33)
SCHEMBL3678165 0.81 CYP1A2 (0.34) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4248245 0.81 GABRA1 (0.33) CYP1A2RXRAPPARGRARG
SCHEMBL1304654 0.75 GABRA1 (0.34) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL3682916 0.70 CYP1A2 (0.34) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL8859880 0.70 MAPT (0.41) TSHRRXRARXRB
SCHEMBL9595008 0.69 GABRA1 (0.33) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL2947022 0.68 PTGS2 (0.47) CYP1A2CYP3A4TSHRRXRAPPARG
SCHEMBL10693024 0.67 GABRA1 (0.34) CYP1A2CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090048408-A1 CATALYST COMPRISING HETEROLEPTIC ALUMINUM AND COBALT COMPOUNDS AND A METHOD OF PREPARING POLYBUTADIENE USING THE SAME KOREA KUMHO PETROCHEMICAL CO., LTD. (KR) 2009-02-19 US claimed
US-20090048408-A1 CATALYST COMPRISING HETEROLEPTIC ALUMINUM AND COBALT COMPOUNDS AND A METHOD OF PREPARING POLYBUTADIENE USING THE SAME KOREA KUMHO PETROCHEMICAL CO., LTD. (KR) 2009-02-19 US disclosed