SCHEMBL4246829

SCHEMBL4246829

NC(=O)OCC(O)C(NC(=O)OCc1cncs1)C(Cc1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 19/20 0.50
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4251958 0.88 CYP3A4 (0.52) CYP3A4TDP1
SCHEMBL893245 0.88 CYP3A4 (0.48) CYP3A4TDP1
SCHEMBL4248671 0.83 CYP3A4 (0.49) CYP3A4
SCHEMBL4253503 0.81 CYP3A4 (0.46) CYP3A4
SCHEMBL4248157 0.81 CYP3A4 (0.48) CYP3A4
SCHEMBL4248623 0.76 CYP3A4 (0.45) CYP3A4
SCHEMBL3015198 0.75 TDP1 (0.48) CYP3A4TDP1
SCHEMBL27738871 0.75 CYP3A4 (0.67) CYP3A4
SCHEMBL27738870 0.75 CYP3A4 (0.67) CYP3A4
SCHEMBL893198 0.75 CYP3A4 (0.55) CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed