SCHEMBL4247397

SCHEMBL4247397

O=C(NCCCN(Cc1ccccc1)C(=O)O)OC(Cc1ccc(-c2ccccn2)cc1)c1scnc1-c1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.39
MLNR O43193 1/20 0.39
NR1I2 O75469 1/20 0.39
SLCO2B1 O94956 1/20 0.39
ABCB11 O95342 1/20 0.39
ABCB1 P08183 1/20 0.39
CCKAR P32238 1/20 0.39
OPRK1 P41145 1/20 0.39
GHSR Q92847 1/20 0.39
SLCO1B3 Q9NPD5 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.39
KCNH2 Q12809 1/20 0.36
PPARG P37231 1/20 0.34
DPP4 P27487 1/20 0.33
MC4R P32245 1/20 0.33
MC5R P33032 1/20 0.33
MC3R P41968 1/20 0.33
ANPEP P15144 1/20 0.33
FAAH O00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943500 0.91 UGT1A1 (0.40) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL9943681 0.74 REN (0.39) OPRK1CYP1A2CYP2D6SMN1; SMN2REN
SCHEMBL4247195 0.69 HDAC3 (0.44) HCAR2CHRNA7ASAH1
SCHEMBL893430 0.68 HDAC3 (0.40) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL4252327 0.68 LTB4R2 (0.53) CYP1A2CYP2D6SMN1; SMN2
SCHEMBL893476 0.68 CYP3A4 (0.45) CYP2D6
SCHEMBL9943670 0.67 CYP3A4 (0.39) CYP2D6SMN1; SMN2REN
SCHEMBL9943809 0.66 CCR6 (0.44) ANPEPCYP2D6SMN1; SMN2REN
SCHEMBL4247398 0.66 CYP3A4 (0.48) CYP2D6
SCHEMBL4248621 0.66 CYP3A4 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP claimed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO claimed