SCHEMBL4247873

SCHEMBL4247873

NC(=O)c1ccc(O)cc1.O=C(O)N1CCC(Cc2ccc(Cl)cc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
MGLL Q99685 2/20 0.48
SPR P35270 1/20 0.47
GRIN2D O15399 3/20 0.46
GRIN3B O60391 3/20 0.46
GRIN1 Q05586 3/20 0.46
GRIN2A Q12879 3/20 0.46
GRIN2B Q13224 3/20 0.46
GRIN2C Q14957 3/20 0.46
GRIN3A Q8TCU5 3/20 0.46
ALDH1A1 P00352 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
ADAMTS5 Q9UNA0 1/20 0.45
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTR2B P41595 1/20 0.44
MAPK14 Q16539 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4239619 0.89 GAA (0.65) GAAGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL4768629 0.89 GAA (0.67) GAA
SCHEMBL27689183 0.88 MAOB (0.54) GAAMGLLSPRGRIN2DGRIN3B
SCHEMBL4243148 0.88 GAA (0.55) GAAGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL4243512 0.88 GAA (0.55) GAAMGLLGRIN2DGRIN3BGRIN1
SCHEMBL4959434 0.86 ALDH1A1 (0.59) MGLLSPRALDH1A1ADAMTS5CYP2C9
SCHEMBL5320493 0.85 GAA (0.49) GAAMGLLSPRGRIN2DGRIN3B
SCHEMBL4250202 0.85 GAA (0.52) GAAMGLLGRIN2DGRIN3BGRIN1
SCHEMBL4241028 0.85 MEN1 (0.53) GAAMGLLGRIN1GRIN2B
SCHEMBL4244568 0.85 GAA (0.52) GAAGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170901-A1 Benzoyl Urea Derivatives RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 2009-07-02 US claimed
EP-1771429-A1 NEW BENZOYL UREA DERIVATIVES RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 2007-04-11 EP claimed
WO-2006010966-A1 NEW BENZOYL UREA DERIVATIVES Richter Gedeon Vegyészeti Gyár Rt. (HU) 2006-02-02 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170901-A1 Benzoyl Urea Derivatives OPRM1, GRIN2C, GRIN3A GAA 3604/4885MGLL 4629/4885SPR 3593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.