SCHEMBL4247930

SCHEMBL4247930

CC(=O)N[C@@H](Cc1ccccc1)C(Cc1cncs1)[C@H](O)[C@H](Cc1ccccc1)OC(N)=O

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.41
CYP3A4 P08684 12/20 0.38
CTRB1 P17538 4/20 0.37
GPR142 Q7Z601 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4247931 1.00 ACACB (0.41) ACACBCYP3A4CTRB1GPR142
SCHEMBL4248616 0.85 CYP3A4 (0.37) CYP3A4GPR142
SCHEMBL4248614 0.85 CYP3A4 (0.37) CYP3A4GPR142
SCHEMBL4252268 0.84 CYP3A4 (0.36) CYP3A4
SCHEMBL4251973 0.84 ACACB (0.42) ACACBCYP3A4CTRB1GPR142
SCHEMBL4251176 0.84 ACACB (0.42) ACACBCYP3A4CTRB1GPR142
SCHEMBL4251971 0.84 ACACB (0.42) ACACBCYP3A4CTRB1GPR142
SCHEMBL15967935 0.83 ACACB (0.39) ACACBCYP3A4
SCHEMBL893121 0.83 ACACB (0.39) ACACBCYP3A4
SCHEMBL4246828 0.81 CYP3A4 (0.52) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed