SCHEMBL4248616

SCHEMBL4248616

NC(=O)O[C@@H](Cc1ccccc1)[C@H](O)C(Cc1cncs1)[C@@H](N)Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.37
TDP1 Q9NUW8 1/20 0.37
GPR142 Q7Z601 7/20 0.36
RAB9A P51151 1/20 0.35
SLC15A1 P46059 1/20 0.35
CTSC P53634 1/20 0.35
PARP15 Q460N3 1/20 0.35
PARP10 Q53GL7 1/20 0.35
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4248614 1.00 CYP3A4 (0.37) CYP3A4TDP1GPR142RAB9ASLC15A1
SCHEMBL4247931 0.85 ACACB (0.41) CYP3A4GPR142
SCHEMBL4247930 0.85 ACACB (0.41) CYP3A4GPR142
SCHEMBL4252268 0.81 CYP3A4 (0.36) CYP3A4
SCHEMBL893582 0.80 SLC6A3 (0.37) CYP3A4TDP1GPR142PARP15PARP10
SCHEMBL4255599 0.80 GPR142 (0.40) CYP3A4TDP1GPR142CTSC
SCHEMBL4399069 0.80 GPR142 (0.40) CYP3A4TDP1GPR142CTSC
SCHEMBL4246828 0.77 CYP3A4 (0.52) CYP3A4TDP1
SCHEMBL893583 0.75 GPR142 (0.43) CYP3A4GPR142
SCHEMBL951450 0.71 CYP1A2 (0.45) CYP3A4TDP1GPR142RAB9APARP15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed