SCHEMBL4249241

SCHEMBL4249241

NS(=O)(=O)CCc1ccncn1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.39
HSP90AA1 P07900 1/20 0.38
P2RX7 Q99572 1/20 0.37
HRH4 Q9H3N8 3/20 0.34
CA2 P00918 4/20 0.33
CA12 O43570 3/20 0.33
CA9 Q16790 3/20 0.33
CA14 Q9ULX7 3/20 0.33
CA1 P00915 2/20 0.33
ALDH1A1 P00352 2/20 0.32
NPC1 O15118 2/20 0.32
KCNH3 Q9ULD8 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CYP1B1 Q16678 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31008661 0.81 P2RX7 (0.37) HSP90AA1P2RX7HRH4ALDH1A1NPC1
SCHEMBL28675951 0.81 P2RX7 (0.37) HSP90AA1P2RX7HRH4ALDH1A1NPC1
SCHEMBL1153882 0.81 HSP90AA1 (0.40) HSP90AA1P2RX7HRH4CA2CA12
SCHEMBL4184428 0.76 HRH1 (0.57) CA2CA1ALDH1A1NPC1RAB9A
Potassium SCHEMBL4063307 0.74 HRH1 (0.55) CA2CA1ALDH1A1NPC1RAB9A
SCHEMBL4063300 0.74 HRH1 (0.55) CA2CA1ALDH1A1NPC1RAB9A
SCHEMBL1661146 0.74
SCHEMBL16399930 0.74
SCHEMBL28629862 0.74 KMT2A (0.63) ALDH1A1NPC1RAB9AKMT2AMEN1
SCHEMBL29924865 0.74 KMT2A (0.63) ALDH1A1NPC1RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049494-A2 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP claimed
WO-2008008310-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2008-01-17 WO claimed
EP-2049494-A2 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2009-04-22 EP disclosed
WO-2008008310-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2008-01-17 WO disclosed
EP-1735284-A1 N-(1-ARYLPYRAZOL-4L)SULFONAMIDES AND THEIR USE AS PARASITICIDES Pfizer Limited (GB) 2006-12-27 EP disclosed
WO-2005090313-A1 N-(1-ARYLPYRAZOL-4L)SULFONAMIDES AND THEIR USE AS PARASITICIDES PFIZER LIMITED (GB) 2005-09-29 WO disclosed