SCHEMBL4249698

SCHEMBL4249698

CN(C)c1ccc(N2C(=O)c3ccc(Br)cc3C2=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.67
ESR2 Q92731 2/20 0.67
STAT3 P40763 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
ALDH1A1 P00352 3/20 0.50
POLB P06746 3/20 0.47
RAB9A P51151 2/20 0.46
NPC1 O15118 2/20 0.46
TSHR P16473 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MEN1 O00255 2/20 0.45
GAA P10253 2/20 0.45
KMT2A Q03164 2/20 0.45
CA9 Q16790 3/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 1/20 0.41
APAF1 O14727 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4254027 0.87 ALDH1A1 (0.66) ESR1ESR2NPSR1ALDH1A1POLB
SCHEMBL4257840 0.84 ESR1 (0.73) ESR1ESR2ALDH1A1POLBRAB9A
SCHEMBL4256256 0.83 CA9 (0.61) ESR1ESR2NPSR1ALDH1A1POLB
SCHEMBL4256208 0.81 ALDH1A1 (0.50) ESR1ESR2ALDH1A1POLBRAB9A
SCHEMBL4255818 0.81 MEN1 (0.53) ESR1ESR2ALDH1A1POLBRAB9A
SCHEMBL4252597 0.80 KMT2A (0.67) NPSR1ALDH1A1RAB9AMEN1GAA
SCHEMBL4258439 0.79 ESR1 (0.61) ESR1ALDH1A1MEN1GAAKMT2A
SCHEMBL17946664 0.79 CA9 (0.54) ESR1ESR2NPSR1ALDH1A1RAB9A
SCHEMBL9566633 0.79 ESR1 (0.73) ESR1ESR2STAT3NPSR1ALDH1A1
SCHEMBL5104501 0.78 ESR1 (0.72) ESR1ESR2STAT3NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed