SCHEMBL4251397

SCHEMBL4251397

COC(=O)Cc1cnc[nH]1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
CYP3A4 P08684 2/20 0.61
GABRA1 P14867 1/20 0.61
TSHR P16473 1/20 0.61
NFKB1 P19838 1/20 0.61
GABRR1 P24046 1/20 0.61
GABRR2 P28476 1/20 0.61
GABRA5 P31644 1/20 0.61
GABRB2 P47870 1/20 0.61
GABRA4 P48169 1/20 0.61
KDM4E B2RXH2 2/20 0.59
PMP22 Q01453 2/20 0.59
MAPT P10636 2/20 0.59
QPCT Q16769 1/20 0.51
QPCTL Q9NXS2 1/20 0.51
PKM P14618 1/20 0.48
POLB P06746 2/20 0.48
RECQL P46063 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MEN1 O00255 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31377271 0.82 ALDH1A1 (0.58) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL27475925 0.82 ALDH1A1 (0.58) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL6932429 0.82 QPCT (0.57) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL1387582 0.81 ALDH1A1 (0.56) ALDH1A1CYP3A4GABRA1TSHRNFKB1
Methyl Alcohol SCHEMBL11465646 0.79 ALDH1A1 (0.68) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL890227 0.79
SCHEMBL8818280 0.78 CYP3A4 (0.73) ALDH1A1CYP3A4GABRA1TSHRNFKB1
SCHEMBL29902874 0.78 ALDH1A1 (0.61) ALDH1A1CYP3A4GABRA1TSHRNFKB1
Imidazole Acetic Acid SCHEMBL49 0.76
SCHEMBL8918572 0.76 ALDH1A1 (0.63) ALDH1A1CYP3A4GABRA1TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083816-A2 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS Brystol-Myers Squibb Company (US) 2009-08-05 EP disclosed
WO-2008057775-A2 HETEROCYCLIC AMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-15 WO disclosed
US-5811445-A ANGIOTENSIN II INHIBITORS ROUSSEL UCLAF (FR) 1998-09-22 US disclosed
EP-0836383-A1 COMBINATIONS OF INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1998-04-22 EP disclosed